# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4097778 | 16h | IC50 | > | 10 | uM | ALA4884602 | Not Active | nM | Mus musculus | ||
2. | ALA4549667 | EUB0000720 | IC50 | 100 | nM | ALA4884602 | Active | nM | Mus musculus | |||
3. | ALA4088216 | 14 | IC50 | 4200 | nM | ALA4884602 | Active | nM | Mus musculus | |||
4. | ALA4785812 | 29 | INH | 0 | ALA4667087 | Not Active | % | Mus musculus | ||||
5. | ALA4850219 | (S)-SZM-777 | INH | 0 | ALA4822739 | Active | % | Mus musculus | ||||
6. | ALA4869920 | (R)-SZM-777 | INH | 0 | ALA4822739 | Active | % | Mus musculus | ||||
7. | ALA4860842 | SZM-777 | INH | = | 100 | % | ALA4822739 | % | Mus musculus | |||
8. | ALA4850219 | (S)-SZM-777 | INH | 0 | ALA4822738 | Active | % | Mus musculus | ||||
9. | ALA4869920 | (R)-SZM-777 | INH | 0 | ALA4822738 | Active | % | Mus musculus | ||||
10. | ALA4860842 | SZM-777 | INH | = | 100 | % | ALA4822738 | % | Mus musculus | |||
11. | Tozasertib | VX-680 | INH | 0 | ALA4048554 | Dose-dependent effect | % | Mus musculus | ||||
12. | ALA4076117 | 118 | INH | < | 50 | % | ALA4048560 | % | Mus musculus | |||
13. | ALA4092326 | 117 | INH | < | 50 | % | ALA4048560 | % | Mus musculus | |||
14. | ALA4064992 | 116 | INH | < | 50 | % | ALA4048560 | % | Mus musculus | |||
15. | ALA4062506 | 115 | INH | < | 50 | % | ALA4048560 | % | Mus musculus | |||
16. | ALA4102896 | 114 | INH | < | 50 | % | ALA4048560 | % | Mus musculus | |||
17. | ALA4059775 | 113 | INH | < | 50 | % | ALA4048560 | % | Mus musculus | |||
18. | ALA4095144 | 112 | INH | < | 50 | % | ALA4048560 | % | Mus musculus | |||
19. | ALA4074679 | 111 | INH | < | 50 | % | ALA4048560 | % | Mus musculus | |||
20. | ALA4077374 | 110 | INH | < | 50 | % | ALA4048560 | % | Mus musculus |