# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5278465 | 33 | IC50 | > | 2 | uM | ALA5252899 | nM | Homo sapiens | |||
2. | ALA5288565 | 29 | IC50 | > | 2 | uM | ALA5252899 | nM | Homo sapiens | |||
3. | ALA5270581 | 18 | IC50 | > | 2 | uM | ALA5252899 | nM | Homo sapiens | |||
4. | ALA4213175 | Fig S3, Cpd 6 | IC50 | > | 2 | uM | ALA5252899 | nM | Homo sapiens | |||
5. | ALA5283398 | Fig 5, Cpd 2 | IC50 | = | 1 | uM | ALA5252709 | 6.00 | nM | Homo sapiens | ||
6. | Staurosporine | 1 (Staurosporine) | Kd | = | 1.3 | nM | ALA5252323 | 8.89 | nM | Homo sapiens | ||
7. | ALA5271697 | 8a | INH | = | 25 | % | ALA5252312 | % | Homo sapiens | |||
8. | ALA5271697 | 8a | deltaTm | = | 3.3 | degrees C | ALA5252301 | degrees C | Homo sapiens | |||
9. | ALA5270781 | 38 | IC50 | = | 1.4 | uM | ALA5252015 | 5.85 | nM | Homo sapiens | ||
10. | ALA5266005 | SCH 727965 | IC50 | = | 1 | nM | ALA5250744 | 9.00 | nM | Homo sapiens | ||
11. | roniciclib | RONICICLIB | IC50 | = | 9 | nM | ALA5250744 | 8.05 | nM | Homo sapiens | ||
12. | LY2857785 | 51; LY2857785 | IC50 | = | 400 | nM | ALA5250744 | 6.40 | nM | Homo sapiens | ||
13. | LDC 000067 | 5, LDC000067 | IC50 | > | 2000 | nM | ALA5250744 | nM | Homo sapiens | |||
14. | ALA3673434 | BDBM164883 | IC50 | = | 2460 | nM | ALA5250744 | 5.61 | nM | Homo sapiens | ||
15. | ALA4560679 | BAY-1143572 | IC50 | = | 1000 | nM | ALA5250744 | 6.00 | nM | Homo sapiens | ||
16. | Flavopiridol | 1 | IC50 | = | 170 | nM | ALA5250744 | 6.77 | nM | Homo sapiens | ||
17. | JNJ-7706621 | 3b | IC50 | = | 2 | nM | ALA5246050 | 8.70 | nM | Homo sapiens | ||
18. | ALA5273533 | 37 | INH | = | 91 | % | ALA5244438 | % | Homo sapiens | |||
19. | ALA5281283 | 18 | IC50 | > | 1000 | nM | ALA5244437 | nM | Homo sapiens | |||
20. | CDKI-73 | 12e | INH | 0 | ALA5244107 | Active | % | Homo sapiens |