# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2372311 | 5 | INH | 0 | ALA2434328 | Active | % | Rattus norvegicus | ||||
2. | ALA2372311 | 5 | INH | 0 | ALA2434327 | Active | % | Rattus norvegicus | ||||
3. | ALA2429934 | C9 | INH | 0 | ALA2434326 | Dose-dependent effect | % | Rattus norvegicus | ||||
4. | ALA2429934 | C9 | INH | 0 | ALA2434325 | Active | % | Rattus norvegicus | ||||
5. | ALA2429934 | C9 | INH | = | 70 | % | ALA2434324 | % | Rattus norvegicus | |||
6. | ALA2429934 | C9 | INH | = | 25 | % | ALA2433154 | % | Rattus norvegicus | |||
7. | L-368,899 hydrochloride | 5 | IC50 | = | 370 | nM | ALA2394481 | 6.43 | nM | Rattus norvegicus | ||
8. | ALA2391300 | 1 | IC50 | = | 320 | nM | ALA2394481 | 6.50 | nM | Rattus norvegicus | ||
9. | conivaptan | Conivaptan | Ki | = | 0.48 | nM | ALA4201576 | 9.32 | nM | Rattus norvegicus | ||
10. | ALA1774016 | 40 | pKi | = | 6.71 | ALA1776932 | 6.71 | nM | Rattus norvegicus | |||
11. | ALA1774017 | 41 | pKi | = | 6.69 | ALA1776932 | 6.69 | nM | Rattus norvegicus | |||
12. | ALA1774018 | 42 | pKi | < | 6 | ALA1776932 | nM | Rattus norvegicus | ||||
13. | ALA1774019 | 43 | pKi | = | 6.42 | ALA1776932 | 6.42 | nM | Rattus norvegicus | |||
14. | ALA1774020 | 44 | pKi | < | 6 | ALA1776932 | nM | Rattus norvegicus | ||||
15. | ALA1774021 | 45 | pKi | = | 6.88 | ALA1776932 | 6.88 | nM | Rattus norvegicus | |||
16. | ALA1774022 | 46 | pKi | = | 7.26 | ALA1776932 | 7.26 | nM | Rattus norvegicus | |||
17. | ALA1774023 | 47 | pKi | = | 7.66 | ALA1776932 | 7.66 | nM | Rattus norvegicus | |||
18. | ALA1774024 | 48 | pKi | = | 8.38 | ALA1776932 | 8.38 | nM | Rattus norvegicus | |||
19. | ALA1774014 | 38 | pKi | <= | 5.5 | ALA1776934 | nM | Rattus norvegicus | ||||
20. | ALA1817770 | 68 | pEC50 | = | 7.24 | ALA1819845 | 7.24 | nM | Rattus norvegicus |