# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4095125 | 25 | pIC50 | = | 7.7 | ALA4052574 | 7.70 | nM | Mus musculus | |||
2. | ALA4078601 | 24 | pIC50 | = | 7.9 | ALA4052574 | 7.90 | nM | Mus musculus | |||
3. | ALA4102883 | 23 | pIC50 | = | 6.2 | ALA4052574 | 6.20 | nM | Mus musculus | |||
4. | Ziritaxestat (GLPG1690) | 32; GLPG1690 | INH | 0 | ALA4051890 | Dose-dependent effect | % | Mus musculus | ||||
5. | Ziritaxestat (GLPG1690) | 32; GLPG1690 | IC50 | = | 418 | nM | ALA4051890 | 6.38 | nM | Mus musculus | ||
6. | ALA4086545 | 8h | IC50 | = | 0.2 | uM | ALA4049299 | 6.70 | nM | Mus musculus | ||
7. | PF-8380 | SID174006268 | IC50 | = | 1.7 | nM | ALA4049310 | 8.77 | nM | Mus musculus | ||
8. | PF-8380 | SID174006268 | IC50 | = | 2.8 | nM | ALA4049309 | 8.55 | nM | Mus musculus | ||
9. | ALA4079494 | 21 | IC50 | = | 4 | uM | ALA4049299 | 5.40 | nM | Mus musculus | ||
10. | ALA4084867 | 18 | IC50 | = | 0.5 | uM | ALA4049299 | 6.30 | nM | Mus musculus | ||
11. | ALA4074600 | 8m | IC50 | = | 2 | uM | ALA4049299 | 5.70 | nM | Mus musculus | ||
12. | ALA4083130 | 8j | IC50 | = | 0.2 | uM | ALA4049299 | 6.70 | nM | Mus musculus | ||
13. | ALA4078700 | 8f | IC50 | = | 0.3 | uM | ALA4049299 | 6.52 | nM | Mus musculus | ||
14. | ALA4094307 | 8b | IC50 | = | 0.2 | uM | ALA4049299 | 6.70 | nM | Mus musculus | ||
15. | inhibitor 32 | 32; GK442 | IC50 | = | 0.06 | uM | ALA4049298 | 7.22 | nM | Mus musculus | ||
16. | ALA4075039 | 28b | IC50 | > | 5 | uM | ALA4049298 | nM | Mus musculus | |||
17. | ALA4094633 | 28a; GK400 | IC50 | = | 0.05 | uM | ALA4049298 | 7.30 | nM | Mus musculus | ||
18. | ALA4074111 | 24e | IC50 | > | 5 | uM | ALA4049298 | nM | Mus musculus | |||
19. | ALA4062177 | 24d | IC50 | = | 4.5 | uM | ALA4049298 | 5.35 | nM | Mus musculus | ||
20. | ALA4083902 | 24c | IC50 | > | 5 | uM | ALA4049298 | nM | Mus musculus |