# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4762311 | 18; PPA | IC50(app) | = | 75 | uM | ALA4736579 | 4.12 | nM | Homo sapiens | ||
2. | Ponatinib (AP24534) | 20g, AP24534 | Kd apparent | > | 30000 | nM | ALA3991854 | Inactive | nM | Homo sapiens | ||
3. | Binimetinib | SID174006430 | Kd apparent | > | 30000 | nM | ALA3991854 | Inactive | nM | Homo sapiens | ||
4. | BMS-690514 | BMS-690514 | Kd apparent | > | 30000 | nM | ALA3991854 | Inactive | nM | Homo sapiens | ||
5. | Bafetinib (INNO-406) | 9b | Kd apparent | > | 30000 | nM | ALA3991854 | Inactive | nM | Homo sapiens | ||
6. | X-376 | 2, X376 | Kd apparent | > | 30000 | nM | ALA3991854 | Inactive | nM | Homo sapiens | ||
7. | tesevatinib | TESEVATINIB | Kd apparent | > | 30000 | nM | ALA3991854 | Inactive | nM | Homo sapiens | ||
8. | ALA91829 | 1 | Kd apparent | > | 30000 | nM | ALA3991854 | Inactive | nM | Homo sapiens | ||
9. | ALA1952329 | Table 2, R1C3 | Kd apparent | > | 30000 | nM | ALA3991854 | Inactive | nM | Homo sapiens | ||
10. | PDGFR Tyrosine Kinase Inhibitor VI, SU6668 | 5b | Kd apparent | > | 30000 | nM | ALA3991854 | Inactive | nM | Homo sapiens | ||
11. | FASUDIL | HA-1077 | Kd apparent | > | 30000 | nM | ALA3991854 | Inactive | nM | Homo sapiens | ||
12. | Fostamatinib (R788) | FOSTAMATINIB | Kd apparent | > | 30000 | nM | ALA3991854 | Inactive | nM | Homo sapiens | ||
13. | AMG-900 | SID137275938 | Kd apparent | > | 30000 | nM | ALA3991854 | Inactive | nM | Homo sapiens | ||
14. | ALA1094408 | 49 | Kd apparent | > | 30000 | nM | ALA3991854 | Inactive | nM | Homo sapiens | ||
15. | R406 (free base) | 5, R-406 | Kd apparent | > | 30000 | nM | ALA3991854 | Inactive | nM | Homo sapiens | ||
16. | MnTMPyP pentachloride | 5 | Kd apparent | > | 30000 | nM | ALA3991854 | Inactive | nM | Homo sapiens | ||
17. | 6-(4-methylpiperazin-1-yl)-N-(5-methyl-1H-pyrazol-3-yl)-2-[(E)-2-phenylethenyl]pyrimidin-4-amine | 14, ENMD-2076 | Kd apparent | > | 30000 | nM | ALA3991854 | Inactive | nM | Homo sapiens | ||
18. | GSK1059615 | GSK-1059615 | Kd apparent | > | 30000 | nM | ALA3991854 | Inactive | nM | Homo sapiens | ||
19. | BI 2536 | 1 | Kd apparent | > | 30000 | nM | ALA3991854 | Inactive | nM | Homo sapiens | ||
20. | PHA-848125 | 28, PHA-848125 | Kd apparent | > | 30000 | nM | ALA3991854 | Inactive | nM | Homo sapiens |