# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BIX 02565 | 24, BIX 02565, eutamer | IC50 | = | 97 | nM | ALA5213146 | 7.01 | nM | Homo sapiens | ||
2. | BI 99179 | 13, BI-99179 | % of inhibition | = | 19 | % | ALA5213852 | % | Homo sapiens | |||
3. | moxonidine | 5 | pIC50 | = | 8.45 | ALA4358952 | 8.45 | nM | Homo sapiens | |||
4. | ALA4467833 | 8a | pIC50 | = | 5.13 | ALA4358952 | 5.13 | nM | Homo sapiens | |||
5. | ALA4483022 | 8b | pIC50 | = | 5.14 | ALA4358952 | 5.14 | nM | Homo sapiens | |||
6. | ALA4546903 | 8c | pIC50 | = | 5.47 | ALA4358952 | 5.47 | nM | Homo sapiens | |||
7. | ALA4439953 | 8d | pIC50 | < | 3 | ALA4358952 | nM | Homo sapiens | ||||
8. | ALA4536304 | 8e | pIC50 | = | 8.09 | ALA4358952 | 8.09 | nM | Homo sapiens | |||
9. | ALA4459090 | 9a | pIC50 | = | 6.19 | ALA4358952 | 6.19 | nM | Homo sapiens | |||
10. | ALA4535472 | 9b | pIC50 | = | 7.54 | ALA4358952 | 7.54 | nM | Homo sapiens | |||
11. | ALA4482861 | 9c | pIC50 | = | 6.74 | ALA4358952 | 6.74 | nM | Homo sapiens | |||
12. | ALA4450506 | 9d | Ki | = | 912 | uM | ALA4358952 | nM | Homo sapiens | |||
13. | ALA4450506 | 9d | pIC50 | = | 3.04 | ALA4358952 | nM | Homo sapiens | ||||
14. | ALA4534152 | 9e | pIC50 | = | 3.22 | ALA4358952 | nM | Homo sapiens | ||||
15. | ALA4469237 | 14c | pIC50 | = | 5.12 | ALA4358952 | 5.12 | nM | Homo sapiens | |||
16. | ALA4438158 | 9j | pIC50 | = | 5.87 | ALA4358952 | 5.87 | nM | Homo sapiens | |||
17. | ALA4434967 | 9k | pIC50 | = | 7.98 | ALA4358952 | 7.98 | nM | Homo sapiens | |||
18. | ALA4438801 | 9x | pIC50 | = | 5.26 | ALA4358952 | 5.26 | nM | Homo sapiens | |||
19. | ALA4590209 | 9z | pIC50 | = | 7.19 | ALA4358952 | 7.19 | nM | Homo sapiens | |||
20. | ALA3546398 | BDBM215805 | Ki | = | 2.8 | nM | ALA3888188 | 8.55 | 379190 | nM | Homo sapiens |