# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BAY 678 | 17, BAY-678 | IC50 | > | 30 | uM | ALA5213827 | nM | Homo sapiens | |||
2. | ALA4166112 | 1 | INH | 0 | ALA4133523 | Not Active | % | Homo sapiens | ||||
3. | ALA4159803 | 2 | INH | 0 | ALA4133523 | Not Active | % | Homo sapiens | ||||
4. | ALA190743 | 4o | IC50 | = | 1 | uM | ALA877333 | 6.00 | nM | Homo sapiens | ||
5. | ALA365134 | 4k | IC50 | = | 10.4 | uM | ALA877333 | 4.98 | nM | Homo sapiens | ||
6. | ALA182348 | 6a | IC50 | 0 | uM | ALA833486 | Inactive | nM | Homo sapiens | |||
7. | ALA275180 | 15b | kinact | 0 | min-1 | ALA820164 | No inactivation | Homo sapiens | ||||
8. | ALA275180 | 15b | Ki | = | 324 | uM | ALA818521 | nM | Homo sapiens | |||
9. | ALA276105 | 13a | kinact | = | 0.091 | min-1 | ALA820163 | min-1 | Homo sapiens | |||
10. | ALA276105 | 13a | Ki | = | 625 | uM | ALA818521 | nM | Homo sapiens | |||
11. | ALA278224 | 10 | K inact | = | 0.006 | min-1 | ALA818527 | min-1 | Homo sapiens | |||
12. | ALA278224 | 10 | Ki | = | 5.6 | uM | ALA818521 | 5.25 | nM | Homo sapiens | ||
13. | ALA16054 | 19b | K inact | = | 0.02 | min-1 | ALA818527 | min-1 | Homo sapiens | |||
14. | ALA16054 | 19b | Ki | = | 49 | uM | ALA818521 | 4.31 | nM | Homo sapiens | ||
15. | ALA16064 | 19a | K inact | = | 0.003 | min-1 | ALA818527 | min-1 | Homo sapiens | |||
16. | ALA16064 | 19a | Ki | = | 50 | uM | ALA818521 | 4.30 | nM | Homo sapiens | ||
17. | ALA16143 | 15a | kinact | = | 0.001 | min-1 | ALA820163 | min-1 | Homo sapiens | |||
18. | ALA16143 | 15a | Ki | = | 93 | uM | ALA818521 | 4.03 | nM | Homo sapiens | ||
19. | ALA274455 | 16a | K inact | 0 | min-1 | ALA818528 | No inactivation | Homo sapiens | ||||
20. | ALA274455 | 16a | Ki | = | 0.27 | uM | ALA818521 | 6.57 | nM | Homo sapiens |