# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4277461 | MBP83-99 | IC50 | = | 87 | nM | ALA4253046 | 7.06 | nM | Homo sapiens | ||
2. | ALA4284706 | (Ahx)6MBP85-99 | IC50 | = | 355 | nM | ALA4253046 | 6.45 | nM | Homo sapiens | ||
3. | ALA4292594 | 5 | IC50 | = | 2901 | nM | ALA4253046 | 5.54 | nM | Homo sapiens | ||
4. | ALA4277461 | MBP83-99 | IC50 | = | 13 | nM | ALA4253045 | 7.89 | nM | Homo sapiens | ||
5. | ALA4284706 | (Ahx)6MBP85-99 | IC50 | = | 13 | nM | ALA4253045 | 7.89 | nM | Homo sapiens | ||
6. | ALA4292594 | 5 | IC50 | = | 56 | nM | ALA4253045 | 7.25 | nM | Homo sapiens | ||
7. | ALA1253321 | (6-DMNA)-RSMAAAAL(open) | IC50 | = | 27 | nM | ALA1253009 | 7.57 | nM | Homo sapiens | ||
8. | ALA1253327 | (4-DAPA)-RSMAAAAL(open) | IC50 | = | 28 | nM | ALA1253009 | 7.55 | nM | Homo sapiens | ||
9. | ALA1253323 | (6-DMNA)-RSMAAAAL(closed) | IC50 | = | 11 | nM | ALA1253009 | 7.96 | nM | Homo sapiens | ||
10. | ALA1253322 | (4-DAPA)-RSMAAAAL(closed) | IC50 | = | 4 | nM | ALA1253009 | 8.40 | nM | Homo sapiens | ||
11. | ALA1253324 | (4-DAPA)-HA | Time | = | 0.6 | nanoseconds | ALA1252972 | nanoseconds | Homo sapiens | |||
12. | ALA1253323 | (6-DMNA)-RSMAAAAL(closed) | Time | = | 0.5 | nanoseconds | ALA1252972 | nanoseconds | Homo sapiens | |||
13. | ALA1253322 | (4-DAPA)-RSMAAAAL(closed) | Time | = | 0.82 | nanoseconds | ALA1252972 | nanoseconds | Homo sapiens | |||
14. | ALA1253323 | (6-DMNA)-RSMAAAAL(closed) | FC | = | 1100 | ALA1252965 | Homo sapiens | |||||
15. | ALA1253323 | (6-DMNA)-RSMAAAAL(closed) | FC | = | 109 | ALA1252969 | Homo sapiens | |||||
16. | ALA1253323 | (6-DMNA)-RSMAAAAL(closed) | FC | = | 239 | ALA1252968 | Homo sapiens | |||||
17. | ALA1253323 | (6-DMNA)-RSMAAAAL(closed) | FC | = | 76 | ALA1252967 | Homo sapiens | |||||
18. | ALA1253323 | (6-DMNA)-RSMAAAAL(closed) | FC | = | 76 | ALA1252966 | Homo sapiens | |||||
19. | ALA1253323 | (6-DMNA)-RSMAAAAL(closed) | Activity | = | 4496 | cps/nM | ALA1253010 | cps/nM | Homo sapiens | |||
20. | ALA1253324 | (4-DAPA)-HA | Activity | = | 578 | cps/nM | ALA1253010 | cps/nM | Homo sapiens |