# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PD184352 (CI-1040) | 1 | Kd | > | 10000 | nM | ALA1908538 | nM | Homo sapiens | |||
2. | Barasertib (AZD1152-HQPA) | 34 | Kd | = | 1500 | nM | ALA1908538 | 5.82 | nM | Homo sapiens | ||
3. | Staurosporine (DMSO solution) | 1 (Staurosporine) | Kd | = | 15 | nM | ALA1908538 | 7.82 | nM | Homo sapiens | ||
4. | Pazopanib | 13 | Kd | = | 2600 | nM | ALA1908538 | 5.58 | nM | Homo sapiens | ||
5. | GW2580 (DMSO solution) | K00591a, Diaminopyrimidine1 | Kd | > | 10000 | nM | ALA1908538 | nM | Homo sapiens | |||
6. | Canertinib (CI-1033) | 18 | Kd | = | 45 | nM | ALA1908538 | 7.35 | nM | Homo sapiens | ||
7. | AT7519 | 33 | Kd | > | 10000 | nM | ALA1908538 | nM | Homo sapiens | |||
8. | Sorafenib | 5 | Kd | > | 10000 | nM | ALA1908538 | nM | Homo sapiens | |||
9. | Nilotinib (AMN-107) | 38 | Kd | = | 500 | nM | ALA1908538 | 6.30 | nM | Homo sapiens | ||
10. | GSK690693 | 3g, GSK-690693 | Kd | > | 10000 | nM | ALA1908538 | nM | Homo sapiens | |||
11. | RAF265 (CHIR-265) | CHIR-265/RAF-265 | Kd | = | 7900 | nM | ALA1908538 | 5.10 | nM | Homo sapiens | ||
12. | Bosutinib Isomer 1, Free Base | 1 (SKI-606) | Kd | = | 3.3 | nM | ALA1908538 | 8.48 | nM | Homo sapiens | ||
13. | MLN8054 | MLN-8054 | Kd | = | 68 | nM | ALA1908538 | 7.17 | nM | Homo sapiens | ||
14. | GSK461364 | GSK-461364A | Kd | > | 10000 | nM | ALA1908538 | nM | Homo sapiens | |||
15. | AST-487 (NVP-AST487) | AST-487 | Kd | = | 30 | nM | ALA1908538 | 7.52 | nM | Homo sapiens | ||
16. | SGX-523 | SGX-523 | Kd | > | 10000 | nM | ALA1908538 | nM | Homo sapiens | |||
17. | Tandutinib (MLN518) | 75 | Kd | > | 10000 | nM | ALA1908538 | nM | Homo sapiens | |||
18. | ALA522892 | 5 | Kd | = | 190 | nM | ALA1908538 | 6.72 | nM | Homo sapiens | ||
19. | Motesanib | AMG-706 | Kd | = | 2200 | nM | ALA1908538 | 5.66 | nM | Homo sapiens | ||
20. | SB-203580 | 9 | Kd | > | 10000 | nM | ALA1908538 | nM | Homo sapiens |