# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1921830 | 33, CAT811 | IC50 | = | 30 | nM | ALA4373321 | 7.52 | nM | Homo sapiens | ||
2. | PD 151746 | 2, PD151746 | Ki | = | 5.33 | uM | ALA3224722 | 5.27 | nM | Homo sapiens | ||
3. | ALA366254 | PD-150606 | Ki | = | 0.37 | uM | ALA3224722 | 6.43 | nM | Homo sapiens | ||
4. | ALA1921836 | 40 | IC50 | = | 28000 | nM | ALA1924666 | 4.55 | nM | Homo sapiens | ||
5. | ALA1921835 | 39 | IC50 | = | 1010 | nM | ALA1924666 | 6.00 | nM | Homo sapiens | ||
6. | ALA1921834 | 38 | IC50 | = | 295 | nM | ALA1924666 | 6.53 | nM | Homo sapiens | ||
7. | ALA1921833 | 37 | IC50 | = | 1100 | nM | ALA1924666 | 5.96 | nM | Homo sapiens | ||
8. | ALA1921832 | 36 | IC50 | = | 180 | nM | ALA1924666 | 6.75 | nM | Homo sapiens | ||
9. | ALA1921831 | 34 | IC50 | = | 700 | nM | ALA1924666 | 6.16 | nM | Homo sapiens | ||
10. | ALA1921830 | 33, CAT811 | IC50 | = | 30 | nM | ALA1924666 | 7.52 | nM | Homo sapiens | ||
11. | ALA1921829 | 32 | IC50 | = | 85 | nM | ALA1924666 | 7.07 | nM | Homo sapiens | ||
12. | ALA1921828 | 31 | IC50 | = | 31000 | nM | ALA1924666 | 4.51 | nM | Homo sapiens | ||
13. | ALA1921827 | 30 | IC50 | = | 850 | nM | ALA1924666 | 6.07 | nM | Homo sapiens | ||
14. | ALA1921826 | H1 | IC50 | = | 2400 | nM | ALA1924666 | 5.62 | nM | Homo sapiens | ||
15. | ALA1921825 | B1 | IC50 | = | 280 | nM | ALA1924666 | 6.55 | nM | Homo sapiens | ||
16. | ALA1921824 | A1 | IC50 | = | 3710 | nM | ALA1924666 | 5.43 | nM | Homo sapiens | ||
17. | Carfilzomib | 2 | INH | 0 | ALA3808089 | Not Active | % | Homo sapiens | ||||
18. | Bortezomib (PS-341) | 15 | INH | 0 | ALA3808089 | Not Active | % | Homo sapiens | ||||
19. | MG-132 (Ethanol Solution) | 5 | Ki | = | 653 | nM | ALA3808087 | 6.18 | nM | Homo sapiens | ||
20. | ALA3804980 | 9 | Ki | = | 1708 | nM | ALA3808087 | 5.77 | nM | Homo sapiens |