| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5306285 | EUB0002235 | delta Tm Staurosporine positive control | = | 1.685 | ALA5304879 | Homo sapiens | |||||
| 2. | ALA5306285 | EUB0002235 | delta Tm | = | -0.559 | ALA5304879 | Not Active | Homo sapiens | ||||
| 3. |  ALA5308262 | EUB0002234 | delta Tm Staurosporine positive control | = | 1.685 | ALA5304775 | Homo sapiens | |||||
| 4. | ALA5308262 | EUB0002234 | delta Tm | = | 0.058 | ALA5304775 | Not Active | Homo sapiens | ||||
| 5. |  ALA5308250 | EUB0002186 | delta Tm Staurosporine positive control | = | 2.888 | ALA5304616 | Homo sapiens | |||||
| 6. | ALA5308250 | EUB0002186 | delta Tm | = | -1.342 | ALA5304616 | Not Active | Homo sapiens | ||||
| 7. |  ALA5306577 | EUB0002354 | delta Tm Staurosporine positive control | = | 2.888 | ALA5304517 | Homo sapiens | |||||
| 8. | ALA5306577 | EUB0002354 | delta Tm | = | -1.08 | ALA5304517 | Not Active | Homo sapiens | ||||
| 9. |  TG 100801 | 12, TG100801 | Kd apparent | > | 30000 | nM | ALA3991714 | Inactive | nM | Homo sapiens | ||
| 10. |  Entrectinib | SID103905026 | Kd apparent | > | 30000 | nM | ALA3991714 | Inactive | nM | Homo sapiens | ||
| 11. |  Y-33075 | 23, Y-39983 | Kd apparent | > | 30000 | nM | ALA3991714 | Inactive | nM | Homo sapiens | ||
| 12. |  PHA-848125 | 28, PHA-848125 | Kd apparent | > | 30000 | nM | ALA3991714 | Inactive | nM | Homo sapiens | ||
| 13. |  Ribociclib | RIBOCICLIB | Kd apparent | = | 12308 | nM | ALA3991714 | 4.91 | Uncertain | nM | Homo sapiens | |
| 14. |  Cediranib | 5, ZD-2171 | Kd apparent | > | 30000 | nM | ALA3991714 | Inactive | nM | Homo sapiens | ||
| 15. |  AT9283 | 16, AT9283 | Kd apparent | > | 30000 | nM | ALA3991714 | Inactive | nM | Homo sapiens | ||
| 16. |  BYL719 | 8, NVP-BYL719 | Kd apparent | > | 30000 | nM | ALA3991714 | Inactive | nM | Homo sapiens | ||
| 17. |  GLPG0634 analogue | SID174006711 | Kd apparent | > | 30000 | nM | ALA3991714 | Inactive | nM | Homo sapiens | ||
| 18. |  Gedatolisib (PF-05212384, PKI-587) | 26, PKI-587 | Kd apparent | > | 30000 | nM | ALA3991714 | Inactive | nM | Homo sapiens | ||
| 19. |  Apatinib | SID124955476 | Kd apparent | > | 30000 | nM | ALA3991714 | Inactive | nM | Homo sapiens | ||
| 20. |  CH4987655 | 24, CH4987655 | Kd apparent | > | 30000 | nM | ALA3991714 | Inactive | nM | Homo sapiens |
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