# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5276110 | 7; [3H]RTI-33 | Bmax | = | 15 | pmol/mg | ALA5240738 | pmol/mg | Mus musculus | |||
2. | ALA5276110 | 7; [3H]RTI-33 | Kd | = | 41 | nM | ALA5240738 | 7.39 | nM | Mus musculus | ||
3. | ALA5175064 | 53 | Activity | 0 | ALA5132115 | NA | Mus musculus | |||||
4. | ALA5175064 | 53 | EC50 | = | 6.5 | uM | ALA5132104 | 5.19 | nM | Mus musculus | ||
5. | ALA5175064 | 53 | EC50 | = | 8.9 | uM | ALA5132103 | 5.05 | nM | Mus musculus | ||
6. | ALA5175064 | 53 | Emax | = | 270 | % | ALA5132102 | % | Mus musculus | |||
7. | ALA5175064 | 53 | Emax | = | 320 | % | ALA5132099 | % | Mus musculus | |||
8. | ALA3884102 | 2.HCl | EC50 | = | 940 | nM | ALA3876615 | 6.03 | nM | Mus musculus | ||
9. | ALA4790638 | 84 | Emax | = | 229 | % | ALA4705842 | % | Mus musculus | |||
10. | RTI-13951-33 | RTI-13951-33 | Emax | = | 535 | % | ALA4705842 | % | Mus musculus | |||
11. | ALA4790638 | 84 | EC50 | = | 942 | nM | ALA4705841 | 6.03 | nM | Mus musculus | ||
12. | RTI-13951-33 | RTI-13951-33 | EC50 | = | 25 | nM | ALA4705841 | 7.60 | nM | Mus musculus | ||
13. | ALA4452474 | 5b | EC50 | = | 535 | nM | ALA4326361 | 6.27 | nM | Mus musculus | ||
14. | (1R,2R)-N-[(2S,3S)-2-amino-3-methylpentyl]-N-[4-(4-propylphenyl)phenyl]-2-pyridin-2-ylcyclopropane-1-carboxamide | 129 | EC50 | = | 1140 | nM | ALA4326361 | 5.94 | nM | Mus musculus |