# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5283559 | 5; SJ43489 | Activity | 0 | ALA5226033 | Not Active | Homo sapiens | |||||
2. | ALA5268757 | 2; SJ34739 | Activity | 0 | ALA5226033 | Not Active | Homo sapiens | |||||
3. | BI 2536 | 1 | % of control | = | 56 | % | ALA5213530 | % | Homo sapiens | |||
4. | ALA5178575 | 28; ARUK3001185 | INH | < | 50 | % | ALA5166977 | % | Homo sapiens | |||
5. | ALA97162 | 26 | Ki | = | 501 | nM | ALA5155889 | 6.30 | nM | Homo sapiens | ||
6. | CAY10571 | 3 | Ki | = | 650 | nM | ALA5155889 | 6.19 | nM | Homo sapiens | ||
7. | Casein Kinase inhibitor A51 | COVC-2297157464 | IC50 | = | 5.3 | nM | ALA5123392 | 8.28 | nM | Homo sapiens | ||
8. | Roscovitine (Seliciclib,CYC202) | Roscovitine | IC50 | = | 49 | uM | ALA4424378 | 4.31 | nM | Homo sapiens | ||
9. | NCC007 | 7b; NCC007 | IC50 | = | 1.8 | uM | ALA4424378 | 5.75 | nM | Homo sapiens | ||
10. | Longdaysin | Longdaysin | IC50 | = | 12 | uM | ALA4424378 | 4.92 | nM | Homo sapiens | ||
11. | NCC007 | 7b; NCC007 | INH | > | 50 | % | ALA4424364 | % | Homo sapiens | |||
12. | NCC007 | 7b; NCC007 | INH | 0 | ALA4424359 | Active | % | Homo sapiens | ||||
13. | Longdaysin | Longdaysin | INH | > | 30 | % | ALA4424359 | % | Homo sapiens | |||
14. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405319 | % | Homo sapiens | |||
15. | ALA4559936 | (+/-)-6 | Activity | = | 5.3 | % | ALA4391274 | % | Homo sapiens | |||
16. | ALA4564973 | 50 | INH | = | 81 | % | ALA4389648 | % | Homo sapiens | |||
17. | ALA4555459 | 43 | INH | = | 62 | % | ALA4389171 | % | Homo sapiens | |||
18. | ALA4545456 | 24 | INH | = | 1.5 | % | ALA4387203 | % | Homo sapiens | |||
19. | Abemaciclib | ABEMACICLIB | INH | = | 4.5 | % | ALA4387203 | % | Homo sapiens | |||
20. | ALA4473365 | 7c | Activity | = | 74 | % | ALA4382452 | % | Homo sapiens |