# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Tazobactam acid | 2 Tazobactam | IC50 | = | 2 | uM | ALA1217813 | 5.70 | nM | Pseudomonas aeruginosa | ||
2. | Sulbactam | 1 | IC50 | = | 3 | uM | ALA1217813 | 5.52 | nM | Pseudomonas aeruginosa | ||
3. | clavulanic acid | Clavulanic acid | IC50 | = | 0.1 | uM | ALA1217813 | 7.00 | nM | Pseudomonas aeruginosa | ||
4. | penicillin G | Benzylpenicillin | Kcat/Km | = | 300 | /mM/s | ALA1217816 | /mM/s | Pseudomonas aeruginosa | |||
5. | penicillin G | Benzylpenicillin | Km | = | 4 | uM | ALA1217815 | nM | Pseudomonas aeruginosa | |||
6. | penicillin G | Benzylpenicillin | Kcat | = | 1.2 | /s | ALA1217815 | /s | Pseudomonas aeruginosa | |||
7. | cefaloridine | cephaloridine | Kcat/Km | = | 150 | /mM/s | ALA1217816 | /mM/s | Pseudomonas aeruginosa | |||
8. | cefaloridine | cephaloridine | Km | = | 8 | uM | ALA1217815 | nM | Pseudomonas aeruginosa | |||
9. | cefaloridine | cephaloridine | Kcat | = | 1.2 | /s | ALA1217815 | /s | Pseudomonas aeruginosa | |||
10. | Imipenem | Imipenem | Kcat | 0 | ALA1217816 | Not Determined | Pseudomonas aeruginosa | |||||
11. | ALA158 | aztreonam | Kcat/Km | = | 280 | /mM/s | ALA1217816 | /mM/s | Pseudomonas aeruginosa | |||
12. | Cefepime | 82(Cefepime) | Kcat/Km | = | 10 | /mM/s | ALA1217816 | /mM/s | Pseudomonas aeruginosa | |||
13. | Cefotaxime acid | cefotaxime | Kcat/Km | = | 290 | /mM/s | ALA1217816 | /mM/s | Pseudomonas aeruginosa | |||
14. | Ceftazidime (containing approximately 10% sodium carbonate) | CAZ | Kcat/Km | = | 47 | /mM/s | ALA1217816 | /mM/s | Pseudomonas aeruginosa | |||
15. | Cefoxitin | Cefoxitin | Kcat/Km | 0 | ALA1217816 | Not Determined | Pseudomonas aeruginosa | |||||
16. | ALA1436 | Cefuroxime | Kcat/Km | = | 73 | /mM/s | ALA1217816 | /mM/s | Pseudomonas aeruginosa | |||
17. | ALA617 | Cephalothin | Kcat/Km | = | 2200 | /mM/s | ALA1217816 | /mM/s | Pseudomonas aeruginosa | |||
18. | Piperacillin | Piperacillin | Kcat/Km | = | 300 | /mM/s | ALA1217816 | /mM/s | Pseudomonas aeruginosa | |||
19. | Imipenem | Imipenem | Km | 0 | ALA1217815 | Not Determined | Pseudomonas aeruginosa | |||||
20. | ALA158 | aztreonam | Km | = | 0.36 | uM | ALA1217815 | nM | Pseudomonas aeruginosa |