# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | grassystatin A | 1 | IC50 | = | 0.8 | nM | ALA2064996 | 9.10 | nM | Homo sapiens | ||
2. | oxazine 89 | 89 | IC50 | > | 200 | uM | ALA2353191 | nM | Homo sapiens | |||
3. | ALA2338554 | 1 | Activity | = | 100 | % | ALA2340455 | % | Homo sapiens | |||
4. | ALA2322896 | 6a, (3S,4S)-6a | IC50 | = | 11 | uM | ALA2330924 | 4.96 | nM | Homo sapiens | ||
5. | ALA2322611 | 12a, (3S,4S)-12a | IC50 | > | 30 | uM | ALA2330924 | nM | Homo sapiens | |||
6. | ALA2322207 | (3S,5R)-12 | IC50 | > | 30 | uM | ALA2329598 | nM | Homo sapiens | |||
7. | ALA2024289 | 3 | IC50 | = | 300 | pM | ALA2027029 | 9.52 | nM | Homo sapiens | ||
8. | VTP-27999 | 41 | INH | < | 10 | % | ALA2027810 | % | Homo sapiens | |||
9. | ALA5184529 | 3 | IC50 | = | 12.04 | nM | ALA5158467 | 7.92 | nM | Homo sapiens | ||
10. | ALA5184180 | 2 | IC50 | = | 100 | nM | ALA5158467 | 7.00 | nM | Homo sapiens | ||
11. | ALA5192597 | 7 | IC50 | = | 104 | nM | ALA5158467 | 6.98 | nM | Homo sapiens | ||
12. | ALA5188873 | 6 | IC50 | = | 187 | nM | ALA5158467 | 6.73 | nM | Homo sapiens | ||
13. | ALA5184970 | 5 | IC50 | = | 105 | nM | ALA5158467 | 6.98 | nM | Homo sapiens | ||
14. | ALA5179569 | 4 | IC50 | = | 120 | nM | ALA5158467 | 6.92 | nM | Homo sapiens | ||
15. | ALA2181022 | 9 | IC50 | = | 0.724 | nM | ALA5158467 | 9.14 | nM | Homo sapiens | ||
16. | ALA2181015 | 2 | IC50 | = | 66 | nM | ALA5158467 | 7.18 | nM | Homo sapiens | ||
17. | ALA296588 | Pepstatin | IC50 | = | 0.446 | nM | ALA5158467 | 9.35 | nM | Homo sapiens | ||
18. | ALA3640116 | BDBM100336 | % Ctrl | 106 | % | ALA4887708 | Not Active | % | Homo sapiens | |||
19. | ALA4588900 | EUB0001182 | % Inhibition of Control Values | -16.8 | % | ALA4882562 | % | Homo sapiens | ||||
20. | ALA3403995 | 23 | IC50 | > | 30 | uM | ALA3406669 | nM | Homo sapiens |