# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Tetrodotoxin | TETRODOTOXIN | Kd | = | 1.8 | nM | ALA4393531 | 8.74 | nM | Rattus norvegicus | ||
2. | 5-[2-[5-chloro-2-[(5-ethoxyquinolin-8-yl)sulfonylamino]phenyl]ethynyl]-4-methoxypyridine-2-carboxylic acid | EUB0001566 | % Inhibition of Control Specific Binding (Mean n=2) | -4.9 | % | ALA4886184 | % | Rattus norvegicus | ||||
3. | ALA3342191 | 9 | % Inhibition of Control Specific Binding (Mean n=2) | 3.3 | % | ALA4883777 | % | Rattus norvegicus | ||||
4. | A-1155463 | 17, A-1155463 | % Inhibition of Control Specific Binding (Mean n=2) | 32.3 | % | ALA4883777 | % | Rattus norvegicus | ||||
5. | ALA4551344 | EUB0000746 | % Inhibition of Control Specific Binding (Mean n=2) | -8.2 | % | ALA4883696 | % | Rattus norvegicus | ||||
6. | ALA4228713 | 22 | % Inhibition of Control Specific Binding (Mean n=2) | -2.3 | % | ALA4883696 | % | Rattus norvegicus | ||||
7. | PF 05105679 | 8, PF-05105679 | % inhibition | 32 | % | ALA4883079 | Not Active | % | Rattus norvegicus | |||
8. | ALA4066040 | 12 | % Inhibition of Control Specific Binding (Mean n=2) | 47.3 | % | ALA4880554 | % | Rattus norvegicus | ||||
9. | ALA4093612 | 13 | % Inhibition of Control Specific Binding (Mean n=2) | 35 | % | ALA4880554 | % | Rattus norvegicus | ||||
10. | ALA4533479 | EUB0000339 | % Inhibition of Control Specific Binding (Mean n=2) | 24.4 | % | ALA4880472 | % | Rattus norvegicus | ||||
11. | A192621 | 38 | % Inhibition of Control Specific Binding (Mean n=2) | 29.1 | % | ALA4880472 | % | Rattus norvegicus | ||||
12. | ALA3931977 | 18 | IC50 | = | 5 | uM | ALA3880171 | 5.30 | nM | Rattus norvegicus | ||
13. | ALA3957374 | 16 | IC50 | < | 5 | uM | ALA3880171 | nM | Rattus norvegicus | |||
14. | ALA3900363 | 15 | IC50 | > | 20 | uM | ALA3880171 | nM | Rattus norvegicus | |||
15. | ALA3890550 | 14 | IC50 | = | 5 | uM | ALA3880171 | 5.30 | nM | Rattus norvegicus | ||
16. | ALA3890289 | 13 | IC50 | < | 5 | uM | ALA3880171 | nM | Rattus norvegicus | |||
17. | ALA3935619 | 12 | IC50 | < | 5 | uM | ALA3880171 | nM | Rattus norvegicus | |||
18. | ALA3984416 | 11 | IC50 | = | 5 | uM | ALA3880171 | 5.30 | nM | Rattus norvegicus | ||
19. | ALA3981916 | 10 | IC50 | > | 20 | uM | ALA3880171 | nM | Rattus norvegicus | |||
20. | ALA3952545 | 9 | IC50 | = | 5 | uM | ALA3880171 | 5.30 | nM | Rattus norvegicus |