# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4635206 | Table 1, R4C2 | Kd | = | 20 | uM | ALA4616363 | 4.70 | nM | Homo sapiens | ||
2. | AMG-900 | SID137275938 | Kd apparent | > | 30000 | nM | ALA3991863 | Inactive | nM | Homo sapiens | ||
3. | LDK378 | 6, LDK378 | Kd apparent | > | 30000 | nM | ALA3991863 | Inactive | nM | Homo sapiens | ||
4. | VX-702 | 5, VX-702 | Kd apparent | > | 30000 | nM | ALA3991863 | Inactive | nM | Homo sapiens | ||
5. | SAR407899 | 14C | Kd apparent | > | 30000 | nM | ALA3991863 | Inactive | nM | Homo sapiens | ||
6. | Cobimetinib | 1, XL518, GDC-0973 | Kd apparent | > | 30000 | nM | ALA3991863 | Inactive | nM | Homo sapiens | ||
7. | Varlitinib | VARLITINIB | Kd apparent | > | 30000 | nM | ALA3991863 | Inactive | nM | Homo sapiens | ||
8. | tesevatinib | TESEVATINIB | Kd apparent | > | 30000 | nM | ALA3991863 | Inactive | nM | Homo sapiens | ||
9. | ALA3545137 | PF-00477736 | Kd apparent | > | 30000 | nM | ALA3991863 | Inactive | nM | Homo sapiens | ||
10. | ALA502835 | 3, BIBF1120 | Kd apparent | > | 30000 | nM | ALA3991863 | Inactive | nM | Homo sapiens | ||
11. | Tandutinib (MLN518) | 75 | Kd apparent | > | 30000 | nM | ALA3991863 | Inactive | nM | Homo sapiens | ||
12. | LY2157299 | GALUNISERTIB | Kd apparent | > | 30000 | nM | ALA3991863 | Inactive | nM | Homo sapiens | ||
13. | ALA608533 | PKC-412 | Kd apparent | > | 30000 | nM | ALA3991863 | Inactive | nM | Homo sapiens | ||
14. | TG100-115 | 6 | Kd apparent | > | 30000 | nM | ALA3991863 | Inactive | nM | Homo sapiens | ||
15. | ALA91829 | 1 | Kd apparent | > | 30000 | nM | ALA3991863 | Inactive | nM | Homo sapiens | ||
16. | Danusertib (PHA-739358) | 9d | Kd apparent | > | 30000 | nM | ALA3991863 | Inactive | nM | Homo sapiens | ||
17. | Icotinib | 12k | Kd apparent | > | 30000 | nM | ALA3991863 | Inactive | nM | Homo sapiens | ||
18. | BEZ235 | SID124898663 | Kd apparent | > | 30000 | nM | ALA3991863 | Inactive | nM | Homo sapiens | ||
19. | MK-8033 | 11r, MK-8033 | Kd apparent | > | 30000 | nM | ALA3991863 | Inactive | nM | Homo sapiens | ||
20. | FASUDIL | HA-1077 | Kd apparent | > | 30000 | nM | ALA3991863 | Inactive | nM | Homo sapiens |