# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Y-33075 | 23, Y-39983 | Kd apparent | > | 30000 | nM | ALA3991810 | Inactive | nM | Homo sapiens | ||
2. | Ulixertinib (BVD-523) | ULIXERTINIB | Kd apparent | > | 30000 | nM | ALA3991810 | Inactive | nM | Homo sapiens | ||
3. | CX-4945 (Silmitasertib) | 25n | Kd apparent | > | 30000 | nM | ALA3991810 | Inactive | nM | Homo sapiens | ||
4. | MnTMPyP pentachloride | 5 | Kd apparent | > | 30000 | nM | ALA3991810 | Inactive | nM | Homo sapiens | ||
5. | TG 100801 | 12, TG100801 | Kd apparent | > | 30000 | nM | ALA3991810 | Inactive | nM | Homo sapiens | ||
6. | Palbociclib | 43(table 3) | Kd apparent | > | 30000 | nM | ALA3991810 | Inactive | nM | Homo sapiens | ||
7. | Trametinib (GSK1120212) | TRAMETINIB | Kd apparent | > | 30000 | nM | ALA3991810 | Inactive | nM | Homo sapiens | ||
8. | PF-3758309 | 1, PF-3758309 | Kd apparent | > | 30000 | nM | ALA3991810 | Inactive | nM | Homo sapiens | ||
9. | Vemurafenib (PLX4032, RG7204) | VEMURAFENIB | Kd apparent | > | 30000 | nM | ALA3991810 | Inactive | nM | Homo sapiens | ||
10. | Lapatinib | GW-572016 | Kd apparent | > | 30000 | nM | ALA3991810 | Inactive | nM | Homo sapiens | ||
11. | Varlitinib | VARLITINIB | Kd apparent | > | 30000 | nM | ALA3991810 | Inactive | nM | Homo sapiens | ||
12. | azd-8186 | 13 | Kd apparent | > | 30000 | nM | ALA3991810 | Inactive | nM | Homo sapiens | ||
13. | Crenolanib (CP-868596) | CRENOLANIB | Kd apparent | > | 30000 | nM | ALA3991810 | Inactive | nM | Homo sapiens | ||
14. | BMS-777607 | 10, BMS-777607 | Kd apparent | > | 30000 | nM | ALA3991810 | Inactive | nM | Homo sapiens | ||
15. | Entrectinib | SID103905026 | Kd apparent | > | 30000 | nM | ALA3991810 | Inactive | nM | Homo sapiens | ||
16. | AZD2014 | 21, AZD2014 | Kd apparent | > | 30000 | nM | ALA3991810 | Inactive | nM | Homo sapiens | ||
17. | AZD1208 | 28 | Kd apparent | > | 30000 | nM | ALA3991810 | Inactive | nM | Homo sapiens | ||
18. | Tivozanib (AV-951) | KRN-951 | Kd apparent | > | 30000 | nM | ALA3991810 | Inactive | nM | Homo sapiens | ||
19. | ALA502835 | 3, BIBF1120 | Kd apparent | > | 30000 | nM | ALA3991810 | Inactive | nM | Homo sapiens | ||
20. | LY2603618 | RABUSERTIB | Kd apparent | > | 30000 | nM | ALA3991810 | Inactive | nM | Homo sapiens |