# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PHA-848125 | 28, PHA-848125 | Kd apparent | = | 329 | nM | ALA3991709 | 6.48 | Active | nM | Homo sapiens | |
2. | Afuresertib (GSK2110183) | AFURESERTIB | Kd apparent | > | 30000 | nM | ALA3991709 | Inactive | nM | Homo sapiens | ||
3. | ALA1094408 | 49 | Kd apparent | > | 30000 | nM | ALA3991709 | Inactive | nM | Homo sapiens | ||
4. | Apatinib | SID124955476 | Kd apparent | > | 30000 | nM | ALA3991709 | Inactive | nM | Homo sapiens | ||
5. | omipalisib | SID137275909 | Kd apparent | > | 30000 | nM | ALA3991709 | Inactive | nM | Homo sapiens | ||
6. | TAK-733 | 17, TAK-733 | Kd apparent | > | 30000 | nM | ALA3991709 | Inactive | nM | Homo sapiens | ||
7. | Ribociclib | RIBOCICLIB | Kd apparent | > | 30000 | nM | ALA3991709 | Inactive | nM | Homo sapiens | ||
8. | Brivanib (BMS-540215) | 12 | Kd apparent | > | 30000 | nM | ALA3991709 | Inactive | nM | Homo sapiens | ||
9. | Sotrastaurin | 1 | Kd apparent | > | 30000 | nM | ALA3991709 | Inactive | nM | Homo sapiens | ||
10. | Imatinib (STI571) | 1 | Kd apparent | > | 30000 | nM | ALA3991709 | Inactive | nM | Homo sapiens | ||
11. | AC480 (BMS-599626) | 13, BMS-599626 | Kd apparent | > | 30000 | nM | ALA3991709 | Inactive | nM | Homo sapiens | ||
12. | BMS-690514 | BMS-690514 | Kd apparent | > | 30000 | nM | ALA3991709 | Inactive | nM | Homo sapiens | ||
13. | Temsirolimus (CCI-779, NSC 683864) | Temsirolimus | Kd apparent | > | 30000 | nM | ALA3991709 | Inactive | nM | Homo sapiens | ||
14. | ALA413 | Rapamycin | Kd apparent | > | 30000 | nM | ALA3991709 | Inactive | nM | Homo sapiens | ||
15. | AV 412 | SID137276039 | Kd apparent | > | 30000 | nM | ALA3991709 | Inactive | nM | Homo sapiens | ||
16. | ALA522892 | 5 | Kd apparent | > | 30000 | nM | ALA3991709 | Inactive | nM | Homo sapiens | ||
17. | AZD8055 | 10, AZD-8055 | Kd apparent | > | 30000 | nM | ALA3991709 | Inactive | nM | Homo sapiens | ||
18. | Tirbanibulin | 3, KX-01 | Kd apparent | > | 30000 | nM | ALA3991709 | Inactive | nM | Homo sapiens | ||
19. | CX-4945 (Silmitasertib) | 25n | Kd apparent | > | 30000 | nM | ALA3991709 | Inactive | nM | Homo sapiens | ||
20. | Flavopiridol | 1 | Kd apparent | = | 921 | nM | ALA3991709 | 6.04 | Active | nM | Homo sapiens |