# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Temsirolimus (CCI-779, NSC 683864) | Temsirolimus | Kd apparent | > | 30000 | nM | ALA3991712 | Inactive | nM | Homo sapiens | ||
2. | SCIO 469 hydrochloride | SCIO-469 | Kd apparent | > | 30000 | nM | ALA3991712 | Inactive | nM | Homo sapiens | ||
3. | GSK2636771 | SID174006492 | Kd apparent | > | 30000 | nM | ALA3991712 | Inactive | nM | Homo sapiens | ||
4. | Lenvatinib (E7080) | E7080 | Kd apparent | > | 30000 | nM | ALA3991712 | Inactive | nM | Homo sapiens | ||
5. | ALA1822792 | MK-2461 | Kd apparent | > | 30000 | nM | ALA3991712 | Inactive | nM | Homo sapiens | ||
6. | Dasatinib | 2, BMS-354825 | Kd apparent | > | 30000 | nM | ALA3991712 | Inactive | nM | Homo sapiens | ||
7. | Vemurafenib (PLX4032, RG7204) | VEMURAFENIB | Kd apparent | > | 30000 | nM | ALA3991712 | Inactive | nM | Homo sapiens | ||
8. | SNS-032 (BMS-387032) | 21 | Kd apparent | > | 30000 | nM | ALA3991712 | Inactive | nM | Homo sapiens | ||
9. | ALA3182444 | SID174006374 | Kd apparent | > | 30000 | nM | ALA3991712 | Inactive | nM | Homo sapiens | ||
10. | BYL719 | 8, NVP-BYL719 | Kd apparent | > | 30000 | nM | ALA3991712 | Inactive | nM | Homo sapiens | ||
11. | MnTMPyP pentachloride | 5 | Kd apparent | > | 30000 | nM | ALA3991712 | Inactive | nM | Homo sapiens | ||
12. | Pelitinib | EKB-569 | Kd apparent | > | 30000 | nM | ALA3991712 | Inactive | nM | Homo sapiens | ||
13. | Dabrafenib | 7, GSK2118436 | Kd apparent | > | 30000 | nM | ALA3991712 | Inactive | nM | Homo sapiens | ||
14. | Ribociclib | RIBOCICLIB | Kd apparent | > | 30000 | nM | ALA3991712 | Inactive | nM | Homo sapiens | ||
15. | Apatinib | SID124955476 | Kd apparent | > | 30000 | nM | ALA3991712 | Inactive | nM | Homo sapiens | ||
16. | ALA608533 | PKC-412 | Kd apparent | > | 30000 | nM | ALA3991712 | Inactive | nM | Homo sapiens | ||
17. | CX-4945 (Silmitasertib) | 25n | Kd apparent | > | 30000 | nM | ALA3991712 | Inactive | nM | Homo sapiens | ||
18. | PDGFR Tyrosine Kinase Inhibitor VI, SU6668 | 5b | Kd apparent | > | 30000 | nM | ALA3991712 | Inactive | nM | Homo sapiens | ||
19. | Pexmetinib (ARRY-614) | PEXMETINIB | Kd apparent | > | 30000 | nM | ALA3991712 | Inactive | nM | Homo sapiens | ||
20. | Brivanib (BMS-540215) | 12 | Kd apparent | > | 30000 | nM | ALA3991712 | Inactive | nM | Homo sapiens |