# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5185523 | 7h | Activity | 0 | ALA5117749 | Active | Homo sapiens | |||||
2. | ALA5185523 | 7h | Activity | 0 | ALA5117746 | Active | Homo sapiens | |||||
3. | CYT387 | 28 | Kd apparent | > | 30000 | nM | ALA3991885 | Inactive | nM | Homo sapiens | ||
4. | SAR407899 | 14C | Kd apparent | > | 30000 | nM | ALA3991885 | Inactive | nM | Homo sapiens | ||
5. | TAK-285 | 34e, TAK-285 | Kd apparent | > | 30000 | nM | ALA3991885 | Inactive | nM | Homo sapiens | ||
6. | CYC116 | 13, CYC-116 | Kd apparent | > | 30000 | nM | ALA3991885 | Inactive | nM | Homo sapiens | ||
7. | Losmapimod | 10, GW-856553 | Kd apparent | > | 30000 | nM | ALA3991885 | Inactive | nM | Homo sapiens | ||
8. | KW-2449 | KW-2449 | Kd apparent | > | 30000 | nM | ALA3991885 | Inactive | nM | Homo sapiens | ||
9. | BI 2536 | 1 | Kd apparent | > | 30000 | nM | ALA3991885 | Inactive | nM | Homo sapiens | ||
10. | Afuresertib (GSK2110183) | AFURESERTIB | Kd apparent | > | 30000 | nM | ALA3991885 | Inactive | nM | Homo sapiens | ||
11. | CO-1686 (AVL-301) | ROCILETINIB | Kd apparent | > | 30000 | nM | ALA3991885 | Inactive | nM | Homo sapiens | ||
12. | TG02 (Double bond E) | 26h, SB1317/TG02 | Kd apparent | > | 30000 | nM | ALA3991885 | Inactive | nM | Homo sapiens | ||
13. | OSI-930 | OSI-930 | Kd apparent | > | 30000 | nM | ALA3991885 | Inactive | nM | Homo sapiens | ||
14. | GDC-0941 | 17, GDC-0941 | Kd apparent | > | 30000 | nM | ALA3991885 | Inactive | nM | Homo sapiens | ||
15. | PF-562271 | PF-562271 | Kd apparent | > | 30000 | nM | ALA3991885 | Inactive | nM | Homo sapiens | ||
16. | Crizotinib | 14, PF-2341066 | Kd apparent | > | 30000 | nM | ALA3991885 | Inactive | nM | Homo sapiens | ||
17. | Ponatinib (AP24534) | 20g, AP24534 | Kd apparent | > | 30000 | nM | ALA3991885 | Inactive | nM | Homo sapiens | ||
18. | Dinaciclib (SCH727965) | DINACICLIB | Kd apparent | > | 30000 | nM | ALA3991885 | Inactive | nM | Homo sapiens | ||
19. | Vandetanib | 22 | Kd apparent | > | 30000 | nM | ALA3991885 | Inactive | nM | Homo sapiens | ||
20. | Ribociclib | RIBOCICLIB | Kd apparent | > | 30000 | nM | ALA3991885 | Inactive | nM | Homo sapiens |