# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | TG02 (Double bond E) | 26h, SB1317/TG02 | Kd apparent | > | 30000 | nM | ALA3991608 | Inactive | nM | Homo sapiens | ||
2. | Pexidartinib | PEXIDARTINIB | Kd apparent | > | 30000 | nM | ALA3991608 | Inactive | nM | Homo sapiens | ||
3. | Filgotinib (GLPG0634) | SID174006711 | Kd apparent | > | 30000 | nM | ALA3991608 | Inactive | nM | Homo sapiens | ||
4. | MK-1775 | SID103905025 | Kd apparent | > | 30000 | nM | ALA3991608 | Inactive | nM | Homo sapiens | ||
5. | AZD8055 | 10, AZD-8055 | Kd apparent | > | 30000 | nM | ALA3991608 | Inactive | nM | Homo sapiens | ||
6. | GSK2636771 | SID174006492 | Kd apparent | > | 30000 | nM | ALA3991608 | Inactive | nM | Homo sapiens | ||
7. | ALA3545328 | XL-019 | Kd apparent | > | 30000 | nM | ALA3991608 | Inactive | nM | Homo sapiens | ||
8. | GDC-0980 (RG7422) | 2, GDC-0980 | Kd apparent | > | 30000 | nM | ALA3991608 | Inactive | nM | Homo sapiens | ||
9. | CAL-101 | 74, GS-1101, CAL-101 | Kd apparent | > | 30000 | nM | ALA3991608 | Inactive | nM | Homo sapiens | ||
10. | VX-702 | 5, VX-702 | Kd apparent | > | 30000 | nM | ALA3991608 | Inactive | nM | Homo sapiens | ||
11. | SNS-314 | SID103905586 | Kd apparent | > | 30000 | nM | ALA3991608 | Inactive | nM | Homo sapiens | ||
12. | ALA1950289 | 1, CC-930 | Kd apparent | > | 30000 | nM | ALA3991608 | Inactive | nM | Homo sapiens | ||
13. | Axitinib | AG-13736 | Kd apparent | > | 30000 | nM | ALA3991608 | Inactive | nM | Homo sapiens | ||
14. | SAR407899 | 14C | Kd apparent | > | 30000 | nM | ALA3991608 | Inactive | nM | Homo sapiens | ||
15. | Neratinib (HKI-272) | 25o (table 3) | Kd apparent | > | 30000 | nM | ALA3991608 | Inactive | nM | Homo sapiens | ||
16. | DCC-2036 (Rebastinib) | REBASTINIB | Kd apparent | > | 30000 | nM | ALA3991608 | Inactive | nM | Homo sapiens | ||
17. | PDGFR Tyrosine Kinase Inhibitor VI, SU6668 | 5b | Kd apparent | > | 30000 | nM | ALA3991608 | Inactive | nM | Homo sapiens | ||
18. | JANEX-1 | JANEX-1 | Kd apparent | > | 30000 | nM | ALA3991608 | Inactive | nM | Homo sapiens | ||
19. | AZD7762 | AZD-7762 | Kd apparent | > | 30000 | nM | ALA3991608 | Inactive | nM | Homo sapiens | ||
20. | MK-8776 (SCH 900776) | 29 | Kd apparent | > | 30000 | nM | ALA3991608 | Inactive | nM | Homo sapiens |