# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PHA-793887 | 31 | Kd apparent | > | 30000 | nM | ALA3991689 | Inactive | nM | Homo sapiens | ||
2. | JANEX-1 | JANEX-1 | Kd apparent | > | 30000 | nM | ALA3991689 | Inactive | nM | Homo sapiens | ||
3. | AZD2014 | 21, AZD2014 | Kd apparent | > | 30000 | nM | ALA3991689 | Inactive | nM | Homo sapiens | ||
4. | TG02 (Double bond E) | 26h, SB1317/TG02 | Kd apparent | > | 30000 | nM | ALA3991689 | Inactive | nM | Homo sapiens | ||
5. | Cobimetinib | 1, XL518, GDC-0973 | Kd apparent | > | 30000 | nM | ALA3991689 | Inactive | nM | Homo sapiens | ||
6. | Binimetinib | SID174006430 | Kd apparent | > | 30000 | nM | ALA3991689 | Inactive | nM | Homo sapiens | ||
7. | MK-2206 | 17 | Kd apparent | > | 30000 | nM | ALA3991689 | Inactive | nM | Homo sapiens | ||
8. | ALA3109738 | 7, JNJ-26483327 | Kd apparent | > | 30000 | nM | ALA3991689 | Inactive | nM | Homo sapiens | ||
9. | Bafetinib (INNO-406) | 9b | Kd apparent | > | 30000 | nM | ALA3991689 | Inactive | nM | Homo sapiens | ||
10. | TG 100572 | 4 | Kd apparent | > | 30000 | nM | ALA3991689 | Inactive | nM | Homo sapiens | ||
11. | Ravoxertinib | RAVOXERTINIB | Kd apparent | > | 30000 | nM | ALA3991689 | Inactive | nM | Homo sapiens | ||
12. | PDGFR Tyrosine Kinase Inhibitor VI, SU6668 | 5b | Kd apparent | > | 30000 | nM | ALA3991689 | Inactive | nM | Homo sapiens | ||
13. | AZD6482 | AZD-6482 | Kd apparent | > | 30000 | nM | ALA3991689 | Inactive | nM | Homo sapiens | ||
14. | Amuvatinib (MP-470) | AMUVATINIB | Kd apparent | > | 30000 | nM | ALA3991689 | Inactive | nM | Homo sapiens | ||
15. | ALA3120215 | OSI027 | Kd apparent | > | 30000 | nM | ALA3991689 | Inactive | nM | Homo sapiens | ||
16. | Fedratinib (SAR302503, TG101348) | 2, TG101348 | Kd apparent | > | 30000 | nM | ALA3991689 | Inactive | nM | Homo sapiens | ||
17. | CH4987655 | 24, CH4987655 | Kd apparent | > | 30000 | nM | ALA3991689 | Inactive | nM | Homo sapiens | ||
18. | ALA3545137 | PF-00477736 | Kd apparent | > | 30000 | nM | ALA3991689 | Inactive | nM | Homo sapiens | ||
19. | AZD1152 | 5 | Kd apparent | > | 30000 | nM | ALA3991689 | Inactive | nM | Homo sapiens | ||
20. | Hydroxyfasudil | hydroxyfasudil | Kd apparent | > | 30000 | nM | ALA3991689 | Inactive | nM | Homo sapiens |