# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | R 59-022 | K00070, R59022 | IC50 | = | 20 | uM | ALA4419837 | 4.70 | nM | Homo sapiens | ||
2. | ALA267777 | 10 | IC50 | = | 9 | uM | ALA4419837 | 5.05 | nM | Homo sapiens | ||
3. | ALA267777 | 10 | INH | 0 | ALA4419854 | Active | % | Homo sapiens | ||||
4. | ALA267777 | 10 | INH | 0 | ALA4419855 | Active | % | Homo sapiens | ||||
5. | ALA267777 | 10 | INH | 0 | ALA4419856 | Active | % | Homo sapiens | ||||
6. | ALA267777 | 10 | INH | 0 | ALA4419858 | Active | % | Homo sapiens | ||||
7. | ALA267777 | 10 | INH | 0 | ALA4419859 | Active | % | Homo sapiens | ||||
8. | ALA267777 | 10 | INH | 0 | ALA4419860 | Active | % | Homo sapiens | ||||
9. | ALA267777 | 10 | INH | 0 | ALA4419861 | Active | % | Homo sapiens | ||||
10. | ALA267777 | 10 | INH | 0 | ALA4419897 | Active | % | Homo sapiens | ||||
11. | ALA267777 | 10 | INH | 0 | ALA4419898 | Active | % | Homo sapiens | ||||
12. | ALA267777 | 10 | INH | 0 | ALA4419899 | Active | % | Homo sapiens | ||||
13. | ALA267777 | 10 | INH | 0 | ALA4419900 | Active | % | Homo sapiens | ||||
14. | ALA267777 | 10 | INH | 0 | ALA4419901 | Active | % | Homo sapiens | ||||
15. | ALA267777 | 10 | INH | 0 | ALA4419902 | Active | % | Homo sapiens | ||||
16. | R 59-022 | K00070, R59022 | INH | 0 | ALA4419837 | Dose-dependent effect | % | Homo sapiens | ||||
17. | ALA267777 | 10 | INH | 0 | ALA4419837 | Dose-dependent effect | % | Homo sapiens | ||||
18. | ALA267777 | 10 | Activity | = | 10 | % | ALA4419857 | % | Homo sapiens | |||
19. | ALA460018 | 6a | Activity | = | 72 | % | ALA4413386 | % | Homo sapiens | |||
20. | Urapidil | Urapidil | Activity | = | 75 | % | ALA4413386 | % | Homo sapiens |