# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Axitinib | AG-13736 | Kd apparent | > | 30000 | nM | ALA3991692 | Inactive | nM | Homo sapiens | ||
2. | Pimasertib (AS-703026) | PIMASERTIB | Kd apparent | > | 30000 | nM | ALA3991692 | Inactive | nM | Homo sapiens | ||
3. | Afatinib | BIBW-2992 | Kd apparent | > | 30000 | nM | ALA3991692 | Inactive | nM | Homo sapiens | ||
4. | EMD 1214063 | 22 | Kd apparent | > | 30000 | nM | ALA3991692 | Inactive | nM | Homo sapiens | ||
5. | GSK461364 | GSK-461364A | Kd apparent | > | 30000 | nM | ALA3991692 | Inactive | nM | Homo sapiens | ||
6. | OSI-930 | OSI-930 | Kd apparent | > | 30000 | nM | ALA3991692 | Inactive | nM | Homo sapiens | ||
7. | Gedatolisib (PF-05212384, PKI-587) | 26, PKI-587 | Kd apparent | > | 30000 | nM | ALA3991692 | Inactive | nM | Homo sapiens | ||
8. | Varlitinib | VARLITINIB | Kd apparent | > | 30000 | nM | ALA3991692 | Inactive | nM | Homo sapiens | ||
9. | TG 100801 | 12, TG100801 | Kd apparent | > | 30000 | nM | ALA3991692 | Inactive | nM | Homo sapiens | ||
10. | Pexmetinib (ARRY-614) | PEXMETINIB | Kd apparent | > | 30000 | nM | ALA3991692 | Inactive | nM | Homo sapiens | ||
11. | K-252a | 2 (K-252a) | Kd apparent | > | 30000 | nM | ALA3991692 | Inactive | nM | Homo sapiens | ||
12. | TAK-733 | 17, TAK-733 | Kd apparent | > | 30000 | nM | ALA3991692 | Inactive | nM | Homo sapiens | ||
13. | ALA3120215 | OSI027 | Kd apparent | > | 30000 | nM | ALA3991692 | Inactive | nM | Homo sapiens | ||
14. | LDK378 | 6, LDK378 | Kd apparent | > | 30000 | nM | ALA3991692 | Inactive | nM | Homo sapiens | ||
15. | BAY 869766 | REFAMETINIB | Kd apparent | > | 30000 | nM | ALA3991692 | Inactive | nM | Homo sapiens | ||
16. | FASUDIL | HA-1077 | Kd apparent | > | 30000 | nM | ALA3991692 | Inactive | nM | Homo sapiens | ||
17. | BI 2536 | 1 | Kd apparent | > | 30000 | nM | ALA3991692 | Inactive | nM | Homo sapiens | ||
18. | TAK-593 | 24, TAK-593 | Kd apparent | > | 30000 | nM | ALA3991692 | Inactive | nM | Homo sapiens | ||
19. | ALA1822792 | MK-2461 | Kd apparent | > | 30000 | nM | ALA3991692 | Inactive | nM | Homo sapiens | ||
20. | Y-33075 | 23, Y-39983 | Kd apparent | > | 30000 | nM | ALA3991692 | Inactive | nM | Homo sapiens |