# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | HMN-214 | HMN-214 | Kd apparent | > | 30000 | nM | ALA3991605 | Inactive | nM | Homo sapiens | ||
2. | Linifanib (ABT-869) | 17p, ABT-869 | Kd apparent | > | 30000 | nM | ALA3991605 | Inactive | nM | Homo sapiens | ||
3. | AZD8931 (Sapitinib) | 2, AZD8931 | Kd apparent | > | 30000 | nM | ALA3991605 | Inactive | nM | Homo sapiens | ||
4. | ALA3184679 | AZD-4547 | Kd apparent | > | 30000 | nM | ALA3991605 | Inactive | nM | Homo sapiens | ||
5. | Pimasertib (AS-703026) | PIMASERTIB | Kd apparent | > | 30000 | nM | ALA3991605 | Inactive | nM | Homo sapiens | ||
6. | Palbociclib | 43(table 3) | Kd apparent | > | 30000 | nM | ALA3991605 | Inactive | nM | Homo sapiens | ||
7. | CAL-101 | 74, GS-1101, CAL-101 | Kd apparent | > | 30000 | nM | ALA3991605 | Inactive | nM | Homo sapiens | ||
8. | racemic-tofacitinib | CP-690550 | Kd apparent | > | 30000 | nM | ALA3991605 | Inactive | nM | Homo sapiens | ||
9. | MK-8776 (SCH 900776) | 29 | Kd apparent | > | 30000 | nM | ALA3991605 | Inactive | nM | Homo sapiens | ||
10. | ALA3544944 | XL-413 | Kd apparent | > | 30000 | nM | ALA3991605 | Inactive | nM | Homo sapiens | ||
11. | Erlotinib | Tarceva | Kd apparent | > | 30000 | nM | ALA3991605 | Inactive | nM | Homo sapiens | ||
12. | Canertinib (CI-1033) | 18 | Kd apparent | > | 30000 | nM | ALA3991605 | Inactive | nM | Homo sapiens | ||
13. | RGB-286638 | RGB-286638 | Kd apparent | > | 30000 | nM | ALA3991605 | Inactive | nM | Homo sapiens | ||
14. | MK-1775 | SID103905025 | Kd apparent | > | 30000 | nM | ALA3991605 | Inactive | nM | Homo sapiens | ||
15. | Dabrafenib | 7, GSK2118436 | Kd apparent | > | 30000 | nM | ALA3991605 | Inactive | nM | Homo sapiens | ||
16. | AZD6482 | AZD-6482 | Kd apparent | > | 30000 | nM | ALA3991605 | Inactive | nM | Homo sapiens | ||
17. | AC480 (BMS-599626) | 13, BMS-599626 | Kd apparent | > | 30000 | nM | ALA3991605 | Inactive | nM | Homo sapiens | ||
18. | ALA1233528 | VOLASERTIB | Kd apparent | > | 30000 | nM | ALA3991605 | Inactive | nM | Homo sapiens | ||
19. | ALA574737 | UCN-02 | Kd apparent | > | 30000 | nM | ALA3991605 | Inactive | nM | Homo sapiens | ||
20. | Brivanib (BMS-540215) | 12 | Kd apparent | > | 30000 | nM | ALA3991605 | Inactive | nM | Homo sapiens |