# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | AZD5438 | 6 | Kd apparent | > | 30000 | nM | ALA3991627 | Inactive | nM | Homo sapiens | ||
2. | Dabrafenib | 7, GSK2118436 | Kd apparent | > | 30000 | nM | ALA3991627 | Inactive | nM | Homo sapiens | ||
3. | AT9283 | 16, AT9283 | Kd apparent | > | 30000 | nM | ALA3991627 | Inactive | nM | Homo sapiens | ||
4. | Foretinib (GSK1363089) | EXEL-2880/GSK-1363089 | Kd apparent | > | 30000 | nM | ALA3991627 | Inactive | nM | Homo sapiens | ||
5. | Cabozantinib (XL184, BMS-907351) | CABOZANTINIB | Kd apparent | > | 30000 | nM | ALA3991627 | Inactive | nM | Homo sapiens | ||
6. | PF-3758309 | 1, PF-3758309 | Kd apparent | > | 30000 | nM | ALA3991627 | Inactive | nM | Homo sapiens | ||
7. | Defactinib | DEFACTINIB | Kd apparent | > | 30000 | nM | ALA3991627 | Inactive | nM | Homo sapiens | ||
8. | LY2584702 | LY-2584702 | Kd apparent | > | 30000 | nM | ALA3991627 | Inactive | nM | Homo sapiens | ||
9. | Pelitinib | EKB-569 | Kd apparent | > | 30000 | nM | ALA3991627 | Inactive | nM | Homo sapiens | ||
10. | ALA1950289 | 1, CC-930 | Kd apparent | > | 30000 | nM | ALA3991627 | Inactive | nM | Homo sapiens | ||
11. | ripasudil | ripasudil | Kd apparent | > | 30000 | nM | ALA3991627 | Inactive | nM | Homo sapiens | ||
12. | Fedratinib (SAR302503, TG101348) | 2, TG101348 | Kd apparent | > | 30000 | nM | ALA3991627 | Inactive | nM | Homo sapiens | ||
13. | SGX-523 | SGX-523 | Kd apparent | > | 30000 | nM | ALA3991627 | Inactive | nM | Homo sapiens | ||
14. | KW-2449 | KW-2449 | Kd apparent | > | 30000 | nM | ALA3991627 | Inactive | nM | Homo sapiens | ||
15. | 6-(4-methylpiperazin-1-yl)-N-(5-methyl-1H-pyrazol-3-yl)-2-[(E)-2-phenylethenyl]pyrimidin-4-amine | 14, ENMD-2076 | Kd apparent | > | 30000 | nM | ALA3991627 | Inactive | nM | Homo sapiens | ||
16. | ALA3545328 | XL-019 | Kd apparent | > | 30000 | nM | ALA3991627 | Inactive | nM | Homo sapiens | ||
17. | ridaforolimus | RIDAFOROLIMUS | Kd apparent | > | 30000 | nM | ALA3991627 | Inactive | nM | Homo sapiens | ||
18. | AZD7762 | AZD-7762 | Kd apparent | > | 30000 | nM | ALA3991627 | Inactive | nM | Homo sapiens | ||
19. | Canertinib (CI-1033) | 18 | Kd apparent | > | 30000 | nM | ALA3991627 | Inactive | nM | Homo sapiens | ||
20. | Ponatinib (AP24534) | 20g, AP24534 | Kd apparent | > | 30000 | nM | ALA3991627 | Inactive | nM | Homo sapiens |