# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Ponatinib (AP24534) | 20g, AP24534 | Kd apparent | > | 30000 | nM | ALA3991911 | Inactive | nM | Homo sapiens | ||
2. | BYL719 | 8, NVP-BYL719 | Kd apparent | > | 30000 | nM | ALA3991911 | Inactive | nM | Homo sapiens | ||
3. | Lapatinib | GW-572016 | Kd apparent | > | 30000 | nM | ALA3991911 | Inactive | nM | Homo sapiens | ||
4. | CP-724714 | 4 | Kd apparent | > | 30000 | nM | ALA3991911 | Inactive | nM | Homo sapiens | ||
5. | LY2801653 | MERESTINIB | Kd apparent | > | 30000 | nM | ALA3991911 | Inactive | nM | Homo sapiens | ||
6. | AZD1152 | 5 | Kd apparent | > | 30000 | nM | ALA3991911 | Inactive | nM | Homo sapiens | ||
7. | RAF265 (CHIR-265) | CHIR-265/RAF-265 | Kd apparent | > | 30000 | nM | ALA3991911 | Inactive | nM | Homo sapiens | ||
8. | ALA1950289 | 1, CC-930 | Kd apparent | > | 30000 | nM | ALA3991911 | Inactive | nM | Homo sapiens | ||
9. | MLN2480 | SID174006384 | Kd apparent | > | 30000 | nM | ALA3991911 | Inactive | nM | Homo sapiens | ||
10. | Linifanib (ABT-869) | 17p, ABT-869 | Kd apparent | > | 30000 | nM | ALA3991911 | Inactive | nM | Homo sapiens | ||
11. | XL647 | TESEVATINIB | Kd apparent | > | 30000 | nM | ALA3991911 | Inactive | nM | Homo sapiens | ||
12. | R406 (free base) | 5, R-406 | Kd apparent | > | 30000 | nM | ALA3991911 | Inactive | nM | Homo sapiens | ||
13. | PF-04217903 | SID103905666 | Kd apparent | > | 30000 | nM | ALA3991911 | Inactive | nM | Homo sapiens | ||
14. | AZD8055 | 10, AZD-8055 | Kd apparent | > | 30000 | nM | ALA3991911 | Inactive | nM | Homo sapiens | ||
15. | PX-866 | 4, PX-866 | Kd apparent | > | 30000 | nM | ALA3991911 | Inactive | nM | Homo sapiens | ||
16. | Pimasertib (AS-703026) | PIMASERTIB | Kd apparent | > | 30000 | nM | ALA3991911 | Inactive | nM | Homo sapiens | ||
17. | ONO-4059 analogue | ONO-4059-analogue | Kd apparent | > | 30000 | nM | ALA3991911 | Inactive | nM | Homo sapiens | ||
18. | ALA462018 | TCN-P | Kd apparent | > | 30000 | nM | ALA3991911 | Inactive | nM | Homo sapiens | ||
19. | Crizotinib (PF-02341066) | 14, PF-2341066 | Kd apparent | > | 30000 | nM | ALA3991911 | Inactive | nM | Homo sapiens | ||
20. | JNJ-38877605 | SID137276033 | Kd apparent | > | 30000 | nM | ALA3991911 | Inactive | nM | Homo sapiens |