| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  6-piperidin-4-yloxy-2H-isoquinolin-1-one | 14C | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
| 2. |  LY2801653 | MERESTINIB | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
| 3. |  TG100-115 | 6 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
| 4. |  PF-04217903 | SID103905666 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
| 5. |  AMG-900 | SID137275938 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
| 6. |  LY2157299 | GALUNISERTIB | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
| 7. |  BMS-754807 | 9d, BMS-754807 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
| 8. |  6-(4-methylpiperazin-1-yl)-N-(5-methyl-1H-pyrazol-3-yl)-2-[(E)-2-phenylethenyl]pyrimidin-4-amine | 14, ENMD-2076 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
| 9. |  Vatalanib base | 1 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
| 10. |  Voxtalisib (XL765) | VOXTALISIB | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
| 11. |  Savolitinib (AZD6094) | 28 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
| 12. |  ALA3688339 | BDBM166063 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
| 13. |  Fedratinib (SAR302503, TG101348) | 2, TG101348 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
| 14. |  RGB-286638 | RGB-286638 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
| 15. |  ALA1950289 | 1, CC-930 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
| 16. |  AT9283 | 16, AT9283 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
| 17. |  ALA1952329 | Table 2, R1C3 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
| 18. |  Tucatinib (Irbinitinib, ONT-380) | TUCATINIB | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
| 19. |  Amuvatinib (MP-470) | AMUVATINIB | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
| 20. |  TG02 (Double bond E) | 26h, SB1317/TG02 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens |
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