# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | SAR407899 | 14C | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
2. | LY2801653 | MERESTINIB | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
3. | TG100-115 | 6 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
4. | PF-04217903 | SID103905666 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
5. | AMG-900 | SID137275938 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
6. | LY2157299 | GALUNISERTIB | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
7. | BMS-754807 | 9d, BMS-754807 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
8. | 6-(4-methylpiperazin-1-yl)-N-(5-methyl-1H-pyrazol-3-yl)-2-[(E)-2-phenylethenyl]pyrimidin-4-amine | 14, ENMD-2076 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
9. | Vatalanib base | 1 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
10. | Voxtalisib (XL765) | VOXTALISIB | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
11. | Savolitinib (AZD6094) | 28 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
12. | ALA3688339 | BDBM166063 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
13. | Fedratinib (SAR302503, TG101348) | 2, TG101348 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
14. | RGB-286638 | RGB-286638 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
15. | ALA1950289 | 1, CC-930 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
16. | AT9283 | 16, AT9283 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
17. | ALA1952329 | Table 2, R1C3 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
18. | Tucatinib (Irbinitinib, ONT-380) | TUCATINIB | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
19. | Amuvatinib (MP-470) | AMUVATINIB | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens | ||
20. | TG02 (Double bond E) | 26h, SB1317/TG02 | Kd apparent | > | 30000 | nM | ALA3991733 | Inactive | nM | Homo sapiens |