# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | NAcM-OPT | 67; NAcM-OPT | IC50 | = | 0.17 | uM | ALA4836117 | 6.77 | nM | Homo sapiens | ||
2. | ALA4876194 | 40 | IC50 | = | 0.11 | uM | ALA4836117 | 6.96 | nM | Homo sapiens | ||
3. | ALA4876194 | 40 | EC50 | = | 0.3 | uM | ALA4836116 | 6.52 | nM | Homo sapiens | ||
4. | MLN4924 | 2, MLN4924 | INH | 0 | ALA4817665 | Active | % | Homo sapiens | ||||
5. | MLN4924 | 2, MLN4924 | INH | 0 | ALA4817664 | Active | % | Homo sapiens | ||||
6. | ALA4865016 | 7h; SK-464 | Kd | = | 35 | nM | ALA4817663 | 7.46 | nM | Homo sapiens | ||
7. | MLN4924 | 2, MLN4924 | INH | 0 | ALA4817628 | Active | % | Homo sapiens | ||||
8. | MLN4924 | 2, MLN4924 | INH | 0 | ALA4817627 | Active | % | Homo sapiens | ||||
9. | ALA4865016 | 7h; SK-464 | INH | 0 | ALA4817626 | Active | % | Homo sapiens | ||||
10. | ALA4865016 | 7h; SK-464 | INH | 0 | ALA4817625 | Active | % | Homo sapiens | ||||
11. | ALA4865016 | 7h; SK-464 | INH | 0 | ALA4817624 | Active | % | Homo sapiens | ||||
12. | ALA4865016 | 7h; SK-464 | INH | 0 | ALA4817623 | Active | % | Homo sapiens | ||||
13. | ALA4865016 | 7h; SK-464 | INH | 0 | ALA4817622 | Active | % | Homo sapiens | ||||
14. | ALA4865016 | 7h; SK-464 | INH | 0 | ALA4817621 | Active | % | Homo sapiens | ||||
15. | ALA4865016 | 7h; SK-464 | Activity | 0 | ALA4817620 | Active | Homo sapiens | |||||
16. | ALA1461372 | SID14740624 | Activity | 0 | ALA4817620 | Not Active | Homo sapiens | |||||
17. | ALA4865016 | 7h; SK-464 | Activity | 0 | ALA4817619 | Active | Homo sapiens | |||||
18. | ALA1461372 | SID14740624 | Activity | 0 | ALA4817619 | Not Active | Homo sapiens | |||||
19. | ALA4865016 | 7h; SK-464 | Activity | 0 | ALA4817612 | Active | Homo sapiens | |||||
20. | ALA4866253 | 7n | IC50 | = | 326.46 | nM | ALA4817610 | 6.49 | nM | Homo sapiens |