# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4749391 | 17 | IC50 | = | 49 | nM | ALA4704015 | 7.31 | nM | Mus musculus | ||
2. | ALA4755139 | 16 | IC50 | = | 30 | nM | ALA4704015 | 7.52 | nM | Mus musculus | ||
3. | ALA4764430 | 15 | IC50 | = | 29 | nM | ALA4704015 | 7.54 | nM | Mus musculus | ||
4. | ALA4789376 | 14 | IC50 | = | 25 | nM | ALA4704015 | 7.60 | nM | Mus musculus | ||
5. | ALA4756869 | 13 | IC50 | = | 15 | nM | ALA4704015 | 7.82 | nM | Mus musculus | ||
6. | ALA4794014 | 12 | IC50 | = | 19 | nM | ALA4704015 | 7.72 | nM | Mus musculus | ||
7. | ALA4776610 | 11 | IC50 | = | 14 | nM | ALA4704015 | 7.85 | nM | Mus musculus | ||
8. | ALA4742167 | 10 | IC50 | = | 7200 | nM | ALA4704015 | 5.14 | nM | Mus musculus | ||
9. | GLPG4716 | 9; OATD-01 | Ki | = | 26.05 | nM | ALA4704015 | 7.58 | nM | Mus musculus | ||
10. | GLPG4716 | 9; OATD-01 | IC50 | = | 28 | nM | ALA4704015 | 7.55 | nM | Mus musculus | ||
11. | ALA4758240 | 8 | IC50 | = | 5300 | nM | ALA4704015 | 5.28 | nM | Mus musculus | ||
12. | ALA4758850 | 7 | IC50 | = | 27000 | nM | ALA4704015 | 4.57 | nM | Mus musculus | ||
13. | ALA4209364 | 1 | IC50 | = | 1600 | nM | ALA4704015 | 5.80 | nM | Mus musculus | ||
14. | ALA4791640 | 5 | IC50 | = | 1700 | nM | ALA4704015 | 5.77 | nM | Mus musculus | ||
15. | ALA4580568 | 24 | IC50 | = | 87 | nM | ALA4704015 | 7.06 | nM | Mus musculus | ||
16. | ALA4461925 | 30 | IC50 | = | 74 | nM | ALA4704015 | 7.13 | nM | Mus musculus | ||
17. | ALA4640857 | 11; OAT-1441 | IC50 | = | 137 | nM | ALA4704015 | 6.86 | nM | Mus musculus | ||
18. | ALA4206372 | 9 | IC50 | = | 29 | nM | ALA4704015 | 7.54 | nM | Mus musculus | ||
19. | 1-(3-amino-1H-1,2,4-triazol-5-yl)-N-[2-(4-chlorophenyl)ethyl]-N-(2-methylpropyl)piperidin-4-amine | 7f | IC50 | = | 2955 | nM | ALA4704015 | 5.53 | nM | Mus musculus | ||
20. | ALA4549449 | 40 | INH | = | 35 | % | ALA4357693 | % | Mus musculus |