# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | refametinib | REFAMETINIB | Kd apparent | > | 30000 | nM | ALA3991699 | Inactive | nM | Homo sapiens | ||
2. | Crenolanib (CP-868596) | CRENOLANIB | Kd apparent | > | 30000 | nM | ALA3991699 | Inactive | nM | Homo sapiens | ||
3. | TAK-733 | 17, TAK-733 | Kd apparent | > | 30000 | nM | ALA3991699 | Inactive | nM | Homo sapiens | ||
4. | Canertinib (CI-1033) | 18 | Kd apparent | > | 30000 | nM | ALA3991699 | Inactive | nM | Homo sapiens | ||
5. | OSI-930 | OSI-930 | Kd apparent | > | 30000 | nM | ALA3991699 | Inactive | nM | Homo sapiens | ||
6. | Nilotinib (AMN-107) | 38 | Kd apparent | > | 30000 | nM | ALA3991699 | Inactive | nM | Homo sapiens | ||
7. | CP-547632 | 1 | Kd apparent | > | 30000 | nM | ALA3991699 | Inactive | nM | Homo sapiens | ||
8. | CO-1686 (AVL-301) | ROCILETINIB | Kd apparent | > | 30000 | nM | ALA3991699 | Inactive | nM | Homo sapiens | ||
9. | VX 702 | 5, VX-702 | Kd apparent | > | 30000 | nM | ALA3991699 | Inactive | nM | Homo sapiens | ||
10. | BGT-226 | 53, BGT226 | Kd apparent | > | 30000 | nM | ALA3991699 | Inactive | nM | Homo sapiens | ||
11. | Apatinib | SID124955476 | Kd apparent | > | 30000 | nM | ALA3991699 | Inactive | nM | Homo sapiens | ||
12. | Erlotinib | Tarceva | Kd apparent | > | 30000 | nM | ALA3991699 | Inactive | nM | Homo sapiens | ||
13. | BMS 911543 | BMS-911543 | Kd apparent | > | 30000 | nM | ALA3991699 | Inactive | nM | Homo sapiens | ||
14. | PH-797804 | 9, PH 797804 | Kd apparent | > | 30000 | nM | ALA3991699 | Inactive | nM | Homo sapiens | ||
15. | AZD2014 | 21, AZD2014 | Kd apparent | > | 30000 | nM | ALA3991699 | Inactive | nM | Homo sapiens | ||
16. | Baricitinib | BARICITINIB | Kd apparent | > | 30000 | nM | ALA3991699 | Inactive | nM | Homo sapiens | ||
17. | Alisertib (MLN8237) | 9, MLN-8237 | Kd apparent | > | 30000 | nM | ALA3991699 | Inactive | nM | Homo sapiens | ||
18. | XL147 | SID174006505 | Kd apparent | > | 30000 | nM | ALA3991699 | Inactive | nM | Homo sapiens | ||
19. | Sunitinib | 12b | Kd apparent | > | 30000 | nM | ALA3991699 | Inactive | nM | Homo sapiens | ||
20. | SGX-523 | SGX-523 | Kd apparent | > | 30000 | nM | ALA3991699 | Inactive | nM | Homo sapiens |