# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Lapatinib | GW-572016 | Kd apparent | > | 30000 | nM | ALA3991864 | Inactive | nM | Homo sapiens | ||
2. | LDK378 | 6, LDK378 | Kd apparent | > | 30000 | nM | ALA3991864 | Inactive | nM | Homo sapiens | ||
3. | ALA3545137 | PF-00477736 | Kd apparent | > | 30000 | nM | ALA3991864 | Inactive | nM | Homo sapiens | ||
4. | Barasertib (AZD1152-HQPA) | 34 | Kd apparent | > | 30000 | nM | ALA3991864 | Inactive | nM | Homo sapiens | ||
5. | Varlitinib | VARLITINIB | Kd apparent | > | 30000 | nM | ALA3991864 | Inactive | nM | Homo sapiens | ||
6. | AMG-900 | SID137275938 | Kd apparent | > | 30000 | nM | ALA3991864 | Inactive | nM | Homo sapiens | ||
7. | Defactinib | DEFACTINIB | Kd apparent | > | 30000 | nM | ALA3991864 | Inactive | nM | Homo sapiens | ||
8. | Sotrastaurin | 1 | Kd apparent | > | 30000 | nM | ALA3991864 | Inactive | nM | Homo sapiens | ||
9. | CH4987655 | 24, CH4987655 | Kd apparent | > | 30000 | nM | ALA3991864 | Inactive | nM | Homo sapiens | ||
10. | ALA3120215 | OSI027 | Kd apparent | > | 30000 | nM | ALA3991864 | Inactive | nM | Homo sapiens | ||
11. | Bafetinib (INNO-406) | 9b | Kd apparent | > | 30000 | nM | ALA3991864 | Inactive | nM | Homo sapiens | ||
12. | Pexidartinib | PEXIDARTINIB | Kd apparent | > | 30000 | nM | ALA3991864 | Inactive | nM | Homo sapiens | ||
13. | ALA91829 | 1 | Kd apparent | > | 30000 | nM | ALA3991864 | Inactive | nM | Homo sapiens | ||
14. | ALA3699142 | BDBM142744 | Kd apparent | > | 30000 | nM | ALA3991864 | Inactive | nM | Homo sapiens | ||
15. | BMS-690514 | BMS-690514 | Kd apparent | > | 30000 | nM | ALA3991864 | Inactive | nM | Homo sapiens | ||
16. | Tivozanib (AV-951) | KRN-951 | Kd apparent | > | 30000 | nM | ALA3991864 | Inactive | nM | Homo sapiens | ||
17. | racemic-tofacitinib | CP-690550 | Kd apparent | > | 30000 | nM | ALA3991864 | Inactive | nM | Homo sapiens | ||
18. | CAL-101 | 74, GS-1101, CAL-101 | Kd apparent | > | 30000 | nM | ALA3991864 | Inactive | nM | Homo sapiens | ||
19. | Golvatinib (E7050) | GOLVATINIB | Kd apparent | > | 30000 | nM | ALA3991864 | Inactive | nM | Homo sapiens | ||
20. | MK-8033 | 11r, MK-8033 | Kd apparent | > | 30000 | nM | ALA3991864 | Inactive | nM | Homo sapiens |