# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | AMG-208 | 4 | Kd apparent | > | 30000 | nM | ALA3991883 | Inactive | nM | Homo sapiens | ||
2. | avutometinib | 1, CH5126766/RO5126766 | Kd apparent | > | 30000 | nM | ALA3991883 | Inactive | nM | Homo sapiens | ||
3. | Ibrutinib (PCI-32765) | SID124898784 | Kd apparent | > | 30000 | nM | ALA3991883 | Inactive | nM | Homo sapiens | ||
4. | ripasudil | ripasudil | Kd apparent | > | 30000 | nM | ALA3991883 | Inactive | nM | Homo sapiens | ||
5. | Fostamatinib (R788) | FOSTAMATINIB | Kd apparent | > | 30000 | nM | ALA3991883 | Inactive | nM | Homo sapiens | ||
6. | CYC116 | 13, CYC-116 | Kd apparent | > | 30000 | nM | ALA3991883 | Inactive | nM | Homo sapiens | ||
7. | Motesanib | AMG-706 | Kd apparent | > | 30000 | nM | ALA3991883 | Inactive | nM | Homo sapiens | ||
8. | Voxtalisib (XL765) | VOXTALISIB | Kd apparent | > | 30000 | nM | ALA3991883 | Inactive | nM | Homo sapiens | ||
9. | BMS-777607 | 10, BMS-777607 | Kd apparent | > | 30000 | nM | ALA3991883 | Inactive | nM | Homo sapiens | ||
10. | ALA574737 | UCN-02 | Kd apparent | > | 30000 | nM | ALA3991883 | Inactive | nM | Homo sapiens | ||
11. | Cerdulatinib hydrochloride | Cerdulatinib Hydrochloride | Kd apparent | > | 30000 | nM | ALA3991883 | Inactive | nM | Homo sapiens | ||
12. | Axitinib | AG-13736 | Kd apparent | > | 30000 | nM | ALA3991883 | Inactive | nM | Homo sapiens | ||
13. | OSI-930 | OSI-930 | Kd apparent | > | 30000 | nM | ALA3991883 | Inactive | nM | Homo sapiens | ||
14. | glesatinib | MGCD265 | Kd apparent | > | 30000 | nM | ALA3991883 | Inactive | nM | Homo sapiens | ||
15. | SU 14813 | SU-14813 | Kd apparent | > | 30000 | nM | ALA3991883 | Inactive | nM | Homo sapiens | ||
16. | ALA3688339 | BDBM166063 | Kd apparent | > | 30000 | nM | ALA3991883 | Inactive | nM | Homo sapiens | ||
17. | Ravoxertinib | RAVOXERTINIB | Kd apparent | > | 30000 | nM | ALA3991883 | Inactive | nM | Homo sapiens | ||
18. | Pexidartinib | PEXIDARTINIB | Kd apparent | > | 30000 | nM | ALA3991883 | Inactive | nM | Homo sapiens | ||
19. | 6-piperidin-4-yloxy-2H-isoquinolin-1-one | 14C | Kd apparent | > | 30000 | nM | ALA3991883 | Inactive | nM | Homo sapiens | ||
20. | Canertinib (CI-1033) | 18 | Kd apparent | > | 30000 | nM | ALA3991883 | Inactive | nM | Homo sapiens |