# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Ribociclib | RIBOCICLIB | Kd apparent | > | 30000 | nM | ALA3991820 | Inactive | nM | Homo sapiens | ||
2. | LY2157299 | GALUNISERTIB | Kd apparent | > | 30000 | nM | ALA3991820 | Inactive | nM | Homo sapiens | ||
3. | Filgotinib (GLPG0634) | SID174006711 | Kd apparent | > | 30000 | nM | ALA3991820 | Inactive | nM | Homo sapiens | ||
4. | CP-724714 | 4 | Kd apparent | > | 30000 | nM | ALA3991820 | Inactive | nM | Homo sapiens | ||
5. | Hydroxyfasudil | hydroxyfasudil | Kd apparent | > | 30000 | nM | ALA3991820 | Inactive | nM | Homo sapiens | ||
6. | Icotinib | 12k | Kd apparent | > | 30000 | nM | ALA3991820 | Inactive | nM | Homo sapiens | ||
7. | AEE788 (NVP-AEE788) | GNF-Pf-5343 | Kd apparent | > | 30000 | nM | ALA3991820 | Inactive | nM | Homo sapiens | ||
8. | Nilotinib (AMN-107) | 38 | Kd apparent | > | 30000 | nM | ALA3991820 | Inactive | nM | Homo sapiens | ||
9. | SU 14813 | SU-14813 | Kd apparent | > | 30000 | nM | ALA3991820 | Inactive | nM | Homo sapiens | ||
10. | ALA576982 | 7, AC220 | Kd apparent | > | 30000 | nM | ALA3991820 | Inactive | nM | Homo sapiens | ||
11. | SCIO 469 hydrochloride | SCIO-469 | Kd apparent | > | 30000 | nM | ALA3991820 | Inactive | nM | Homo sapiens | ||
12. | Entrectinib | SID103905026 | Kd apparent | > | 30000 | nM | ALA3991820 | Inactive | nM | Homo sapiens | ||
13. | Lapatinib | GW-572016 | Kd apparent | > | 30000 | nM | ALA3991820 | Inactive | nM | Homo sapiens | ||
14. | BMS-754807 | 9d, BMS-754807 | Kd apparent | > | 30000 | nM | ALA3991820 | Inactive | nM | Homo sapiens | ||
15. | BKM120 | 15, NVP-BKM120 | Kd apparent | > | 30000 | nM | ALA3991820 | Inactive | nM | Homo sapiens | ||
16. | Osimertinib (AZD9291) | 8 | Kd apparent | > | 30000 | nM | ALA3991820 | Inactive | nM | Homo sapiens | ||
17. | EOC317 | ACTB-1003 | Kd apparent | > | 30000 | nM | ALA3991820 | Inactive | nM | Homo sapiens | ||
18. | Everolimus | EVEROLIMUS | Kd apparent | > | 30000 | nM | ALA3991820 | Inactive | nM | Homo sapiens | ||
19. | Bosutinib Isomer 1, Free Base | 1 (SKI-606) | Kd apparent | > | 30000 | nM | ALA3991820 | Inactive | nM | Homo sapiens | ||
20. | MK-8033 | 11r, MK-8033 | Kd apparent | > | 30000 | nM | ALA3991820 | Inactive | nM | Homo sapiens |