# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Abemaciclib | ABEMACICLIB | Kd apparent | > | 30000 | nM | ALA3991612 | Inactive | nM | Homo sapiens | ||
2. | Vemurafenib (PLX4032, RG7204) | VEMURAFENIB | Kd apparent | > | 30000 | nM | ALA3991612 | Inactive | nM | Homo sapiens | ||
3. | ALA4084193 | RDEA-436 | Kd apparent | > | 30000 | nM | ALA3991612 | Inactive | nM | Homo sapiens | ||
4. | CH5183284 (Debio-1347) | 8; CH5183284; Debio 1347 | Kd apparent | > | 30000 | nM | ALA3991612 | Inactive | nM | Homo sapiens | ||
5. | Telatinib | BAY-579352 | Kd apparent | > | 30000 | nM | ALA3991612 | Inactive | nM | Homo sapiens | ||
6. | TG 100801 | 12, TG100801 | Kd apparent | > | 30000 | nM | ALA3991612 | Inactive | nM | Homo sapiens | ||
7. | BYL719 | 8, NVP-BYL719 | Kd apparent | > | 30000 | nM | ALA3991612 | Inactive | nM | Homo sapiens | ||
8. | Y-33075 | 23, Y-39983 | Kd apparent | > | 30000 | nM | ALA3991612 | Inactive | nM | Homo sapiens | ||
9. | SNS-032 (BMS-387032) | 21 | Kd apparent | > | 30000 | nM | ALA3991612 | Inactive | nM | Homo sapiens | ||
10. | Tideglusib | TIDEGLUSIB | Kd apparent | > | 30000 | nM | ALA3991612 | Inactive | nM | Homo sapiens | ||
11. | MK-8776 (SCH 900776) | 29 | Kd apparent | > | 30000 | nM | ALA3991612 | Inactive | nM | Homo sapiens | ||
12. | Imatinib (STI571) | 1 | Kd apparent | > | 30000 | nM | ALA3991612 | Inactive | nM | Homo sapiens | ||
13. | CEP-32496 | 40, CEP-32496 | Kd apparent | > | 30000 | nM | ALA3991612 | Inactive | nM | Homo sapiens | ||
14. | Palbociclib | 43(table 3) | Kd apparent | > | 30000 | nM | ALA3991612 | Inactive | nM | Homo sapiens | ||
15. | Sunitinib | 12b | Kd apparent | > | 30000 | nM | ALA3991612 | Inactive | nM | Homo sapiens | ||
16. | AZD8931 (Sapitinib) | 2, AZD8931 | Kd apparent | > | 30000 | nM | ALA3991612 | Inactive | nM | Homo sapiens | ||
17. | K-252a | 2 (K-252a) | Kd apparent | > | 30000 | nM | ALA3991612 | Inactive | nM | Homo sapiens | ||
18. | Entrectinib | SID103905026 | Kd apparent | > | 30000 | nM | ALA3991612 | Inactive | nM | Homo sapiens | ||
19. | GSK1070916 | GSK-1070916 | Kd apparent | > | 30000 | nM | ALA3991612 | Inactive | nM | Homo sapiens | ||
20. | Perifosine (KRX-0401) | OPP | Kd apparent | > | 30000 | nM | ALA3991612 | Inactive | nM | Homo sapiens |