# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | GLPG0634 analogue | SID174006711 | Kd apparent | > | 30000 | nM | ALA3991732 | Inactive | nM | Homo sapiens | ||
2. | TG 100572 | 4 | Kd apparent | > | 30000 | nM | ALA3991732 | Inactive | nM | Homo sapiens | ||
3. | TG 100801 | 12, TG100801 | Kd apparent | > | 30000 | nM | ALA3991732 | Inactive | nM | Homo sapiens | ||
4. | Crenolanib (CP-868596) | CRENOLANIB | Kd apparent | = | 2566 | nM | ALA3991732 | 5.59 | Active | nM | Homo sapiens | |
5. | AZD5438 | 6 | Kd apparent | > | 30000 | nM | ALA3991732 | Inactive | nM | Homo sapiens | ||
6. | Brivanib Alaninate (BMS-582664) | 9 | Kd apparent | > | 30000 | nM | ALA3991732 | Inactive | nM | Homo sapiens | ||
7. | Vatalanib base | 1 | Kd apparent | > | 30000 | nM | ALA3991732 | Inactive | nM | Homo sapiens | ||
8. | Sunitinib | 12b | Kd apparent | > | 30000 | nM | ALA3991732 | Inactive | nM | Homo sapiens | ||
9. | GDC-0941 | 17, GDC-0941 | Kd apparent | > | 30000 | nM | ALA3991732 | Inactive | nM | Homo sapiens | ||
10. | SGX-523 | SGX-523 | Kd apparent | > | 30000 | nM | ALA3991732 | Inactive | nM | Homo sapiens | ||
11. | GSK2636771 | SID174006492 | Kd apparent | > | 30000 | nM | ALA3991732 | Inactive | nM | Homo sapiens | ||
12. | BMS 911543 | BMS-911543 | Kd apparent | > | 30000 | nM | ALA3991732 | Inactive | nM | Homo sapiens | ||
13. | AC480 (BMS-599626) | 13, BMS-599626 | Kd apparent | > | 30000 | nM | ALA3991732 | Inactive | nM | Homo sapiens | ||
14. | SNS-032 (BMS-387032) | 21 | Kd apparent | > | 30000 | nM | ALA3991732 | Inactive | nM | Homo sapiens | ||
15. | Palbociclib | 43(table 3) | Kd apparent | > | 30000 | nM | ALA3991732 | Inactive | nM | Homo sapiens | ||
16. | Temsirolimus (CCI-779, NSC 683864) | Temsirolimus | Kd apparent | > | 30000 | nM | ALA3991732 | Inactive | nM | Homo sapiens | ||
17. | Ulixertinib (BVD-523) | ULIXERTINIB | Kd apparent | > | 30000 | nM | ALA3991732 | Inactive | nM | Homo sapiens | ||
18. | Savolitinib (AZD6094) | 28 | Kd apparent | > | 30000 | nM | ALA3991732 | Inactive | nM | Homo sapiens | ||
19. | ALA3184679 | AZD-4547 | Kd apparent | > | 30000 | nM | ALA3991732 | Inactive | nM | Homo sapiens | ||
20. | TAK-733 | 17, TAK-733 | Kd apparent | > | 30000 | nM | ALA3991732 | Inactive | nM | Homo sapiens |