# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | GSK2636771 | SID174006492 | Kd apparent | > | 30000 | nM | ALA3991617 | Inactive | nM | Homo sapiens | ||
2. | ALA1950289 | 1, CC-930 | Kd apparent | > | 30000 | nM | ALA3991617 | Inactive | nM | Homo sapiens | ||
3. | Dasatinib | 2, BMS-354825 | Kd apparent | > | 30000 | nM | ALA3991617 | Inactive | nM | Homo sapiens | ||
4. | Baricitinib | BARICITINIB | Kd apparent | > | 30000 | nM | ALA3991617 | Inactive | nM | Homo sapiens | ||
5. | AZD6482 | AZD-6482 | Kd apparent | > | 30000 | nM | ALA3991617 | Inactive | nM | Homo sapiens | ||
6. | Dinaciclib (SCH727965) | DINACICLIB | Kd apparent | > | 30000 | nM | ALA3991617 | Inactive | nM | Homo sapiens | ||
7. | Ruxolitinib (INCB018424) | 3, INCB-018424 | Kd apparent | > | 30000 | nM | ALA3991617 | Inactive | nM | Homo sapiens | ||
8. | Lenvatinib (E7080) | E7080 | Kd apparent | > | 30000 | nM | ALA3991617 | Inactive | nM | Homo sapiens | ||
9. | Vemurafenib (PLX4032, RG7204) | VEMURAFENIB | Kd apparent | > | 30000 | nM | ALA3991617 | Inactive | nM | Homo sapiens | ||
10. | CAL-101 | 74, GS-1101, CAL-101 | Kd apparent | > | 30000 | nM | ALA3991617 | Inactive | nM | Homo sapiens | ||
11. | racemic-tofacitinib | CP-690550 | Kd apparent | > | 30000 | nM | ALA3991617 | Inactive | nM | Homo sapiens | ||
12. | CP-724714 | 4 | Kd apparent | > | 30000 | nM | ALA3991617 | Inactive | nM | Homo sapiens | ||
13. | BAY 80-6946 (Copanlisib) | 46, BAY80-6946 | Kd apparent | > | 30000 | nM | ALA3991617 | Inactive | nM | Homo sapiens | ||
14. | Telatinib | BAY-579352 | Kd apparent | > | 30000 | nM | ALA3991617 | Inactive | nM | Homo sapiens | ||
15. | CUDC-101 | 8, CDUC-101 | Kd apparent | > | 30000 | nM | ALA3991617 | Inactive | nM | Homo sapiens | ||
16. | Vatalanib base | 1 | Kd apparent | > | 30000 | nM | ALA3991617 | Inactive | nM | Homo sapiens | ||
17. | Fedratinib (SAR302503, TG101348) | 2, TG101348 | Kd apparent | = | 231 | nM | ALA3991617 | 6.64 | Active | nM | Homo sapiens | |
18. | TAK-733 | 17, TAK-733 | Kd apparent | > | 30000 | nM | ALA3991617 | Inactive | nM | Homo sapiens | ||
19. | SU 14813 | SU-14813 | Kd apparent | > | 30000 | nM | ALA3991617 | Inactive | nM | Homo sapiens | ||
20. | CH5183284 (Debio-1347) | 8; CH5183284; Debio 1347 | Kd apparent | > | 30000 | nM | ALA3991617 | Inactive | nM | Homo sapiens |