# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | SU 14813 | SU-14813 | Kd apparent | > | 30000 | nM | ALA3991619 | Inactive | nM | Homo sapiens | ||
2. | CP-724714 | 4 | Kd apparent | > | 30000 | nM | ALA3991619 | Inactive | nM | Homo sapiens | ||
3. | BAY 80-6946 (Copanlisib) | 46, BAY80-6946 | Kd apparent | > | 30000 | nM | ALA3991619 | Inactive | nM | Homo sapiens | ||
4. | Vatalanib base | 1 | Kd apparent | > | 30000 | nM | ALA3991619 | Inactive | nM | Homo sapiens | ||
5. | Sotrastaurin | 1 | Kd apparent | > | 30000 | nM | ALA3991619 | Inactive | nM | Homo sapiens | ||
6. | CO-1686 (AVL-301) | ROCILETINIB | Kd apparent | > | 30000 | nM | ALA3991619 | Inactive | nM | Homo sapiens | ||
7. | AEE788 (NVP-AEE788) | GNF-Pf-5343 | Kd apparent | > | 30000 | nM | ALA3991619 | Inactive | nM | Homo sapiens | ||
8. | Sunitinib | 12b | Kd apparent | > | 30000 | nM | ALA3991619 | Inactive | nM | Homo sapiens | ||
9. | GDC-0941 | 17, GDC-0941 | Kd apparent | > | 30000 | nM | ALA3991619 | Inactive | nM | Homo sapiens | ||
10. | GSK1059615 | GSK-1059615 | Kd apparent | > | 30000 | nM | ALA3991619 | Inactive | nM | Homo sapiens | ||
11. | Golvatinib (E7050) | GOLVATINIB | Kd apparent | > | 30000 | nM | ALA3991619 | Inactive | nM | Homo sapiens | ||
12. | RO5126766 (CH5126766) | 1, CH5126766/RO5126766 | Kd apparent | > | 30000 | nM | ALA3991619 | Inactive | nM | Homo sapiens | ||
13. | Lestaurtinib | CEP-701 | Kd apparent | > | 30000 | nM | ALA3991619 | Inactive | nM | Homo sapiens | ||
14. | Afatinib | BIBW-2992 | Kd apparent | > | 30000 | nM | ALA3991619 | Inactive | nM | Homo sapiens | ||
15. | CAL-101 | 74, GS-1101, CAL-101 | Kd apparent | > | 30000 | nM | ALA3991619 | Inactive | nM | Homo sapiens | ||
16. | CUDC-101 | 8, CDUC-101 | Kd apparent | > | 30000 | nM | ALA3991619 | Inactive | nM | Homo sapiens | ||
17. | Palbociclib | 43(table 3) | Kd apparent | > | 30000 | nM | ALA3991619 | Inactive | nM | Homo sapiens | ||
18. | ALA522892 | 5 | Kd apparent | > | 30000 | nM | ALA3991619 | Inactive | nM | Homo sapiens | ||
19. | Brivanib Alaninate (BMS-582664) | 9 | Kd apparent | > | 30000 | nM | ALA3991619 | Inactive | nM | Homo sapiens | ||
20. | glesatinib | MGCD265 | Kd apparent | > | 30000 | nM | ALA3991619 | Inactive | nM | Homo sapiens |