# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Axitinib | AG-13736 | Kd apparent | > | 30000 | nM | ALA3991881 | Inactive | nM | Homo sapiens | ||
2. | ALA3688339 | BDBM166063 | Kd apparent | > | 30000 | nM | ALA3991881 | Inactive | nM | Homo sapiens | ||
3. | ALA3545328 | XL-019 | Kd apparent | > | 30000 | nM | ALA3991881 | Inactive | nM | Homo sapiens | ||
4. | Canertinib (CI-1033) | 18 | Kd apparent | > | 30000 | nM | ALA3991881 | Inactive | nM | Homo sapiens | ||
5. | Gilteritinib | GILTERITINIB | Kd apparent | > | 30000 | nM | ALA3991881 | Inactive | nM | Homo sapiens | ||
6. | Fostamatinib (R788) | FOSTAMATINIB | Kd apparent | > | 30000 | nM | ALA3991881 | Inactive | nM | Homo sapiens | ||
7. | ALA1614701 | AZD-6244 | Kd apparent | > | 30000 | nM | ALA3991881 | Inactive | nM | Homo sapiens | ||
8. | AMG-208 | 4 | Kd apparent | > | 30000 | nM | ALA3991881 | Inactive | nM | Homo sapiens | ||
9. | Perifosine (KRX-0401) | OPP | Kd apparent | > | 30000 | nM | ALA3991881 | Inactive | nM | Homo sapiens | ||
10. | AMG-900 | SID137275938 | Kd apparent | > | 30000 | nM | ALA3991881 | Inactive | nM | Homo sapiens | ||
11. | Vandetanib | 22 | Kd apparent | > | 30000 | nM | ALA3991881 | Inactive | nM | Homo sapiens | ||
12. | Neratinib (HKI-272) | 25o (table 3) | Kd apparent | > | 30000 | nM | ALA3991881 | Inactive | nM | Homo sapiens | ||
13. | Tucatinib (Irbinitinib, ONT-380) | TUCATINIB | Kd apparent | > | 30000 | nM | ALA3991881 | Inactive | nM | Homo sapiens | ||
14. | AZD8055 | 10, AZD-8055 | Kd apparent | > | 30000 | nM | ALA3991881 | Inactive | nM | Homo sapiens | ||
15. | Nilotinib (AMN-107) | 38 | Kd apparent | > | 30000 | nM | ALA3991881 | Inactive | nM | Homo sapiens | ||
16. | SCIO 469 hydrochloride | SCIO-469 | Kd apparent | > | 30000 | nM | ALA3991881 | Inactive | nM | Homo sapiens | ||
17. | Savolitinib (AZD6094) | 28 | Kd apparent | > | 30000 | nM | ALA3991881 | Inactive | nM | Homo sapiens | ||
18. | ALA502835 | 3, BIBF1120 | Kd apparent | > | 30000 | nM | ALA3991881 | Inactive | nM | Homo sapiens | ||
19. | DCC-2036 (Rebastinib) | REBASTINIB | Kd apparent | > | 30000 | nM | ALA3991881 | Inactive | nM | Homo sapiens | ||
20. | Poziotinib (HM781-36B) | POZIOTINIB | Kd apparent | > | 30000 | nM | ALA3991881 | Inactive | nM | Homo sapiens |