# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BAY 80-6946 (Copanlisib) | 46, BAY80-6946 | Kd apparent | > | 30000 | nM | ALA3991886 | Inactive | nM | Homo sapiens | ||
2. | Afatinib | BIBW-2992 | Kd apparent | > | 30000 | nM | ALA3991886 | Inactive | nM | Homo sapiens | ||
3. | Ibrutinib (PCI-32765) | SID124898784 | Kd apparent | > | 30000 | nM | ALA3991886 | Inactive | nM | Homo sapiens | ||
4. | PF-3758309 | 1, PF-3758309 | Kd apparent | > | 30000 | nM | ALA3991886 | Inactive | nM | Homo sapiens | ||
5. | TAK-285 | 34e, TAK-285 | Kd apparent | > | 30000 | nM | ALA3991886 | Inactive | nM | Homo sapiens | ||
6. | Axitinib | AG-13736 | Kd apparent | > | 30000 | nM | ALA3991886 | Inactive | nM | Homo sapiens | ||
7. | ALA3182444 | SID174006374 | Kd apparent | > | 30000 | nM | ALA3991886 | Inactive | nM | Homo sapiens | ||
8. | AZD8055 | 10, AZD-8055 | Kd apparent | > | 30000 | nM | ALA3991886 | Inactive | nM | Homo sapiens | ||
9. | OSI-930 | OSI-930 | Kd apparent | > | 30000 | nM | ALA3991886 | Inactive | nM | Homo sapiens | ||
10. | Erlotinib | Tarceva | Kd apparent | > | 30000 | nM | ALA3991886 | Inactive | nM | Homo sapiens | ||
11. | Bafetinib (INNO-406) | 9b | Kd apparent | > | 30000 | nM | ALA3991886 | Inactive | nM | Homo sapiens | ||
12. | Vandetanib | 22 | Kd apparent | > | 30000 | nM | ALA3991886 | Inactive | nM | Homo sapiens | ||
13. | JNJ-38877605 | SID137276033 | Kd apparent | > | 30000 | nM | ALA3991886 | Inactive | nM | Homo sapiens | ||
14. | Canertinib (CI-1033) | 18 | Kd apparent | > | 30000 | nM | ALA3991886 | Inactive | nM | Homo sapiens | ||
15. | GDC-0941 | 17, GDC-0941 | Kd apparent | > | 30000 | nM | ALA3991886 | Inactive | nM | Homo sapiens | ||
16. | ASP3026 | ASP-3026 | Kd apparent | > | 30000 | nM | ALA3991886 | Inactive | nM | Homo sapiens | ||
17. | ALA3184679 | AZD-4547 | Kd apparent | > | 30000 | nM | ALA3991886 | Inactive | nM | Homo sapiens | ||
18. | ALA1950289 | 1, CC-930 | Kd apparent | > | 30000 | nM | ALA3991886 | Inactive | nM | Homo sapiens | ||
19. | Vatalanib base | 1 | Kd apparent | > | 30000 | nM | ALA3991886 | Inactive | nM | Homo sapiens | ||
20. | JANEX-1 | JANEX-1 | Kd apparent | > | 30000 | nM | ALA3991886 | Inactive | nM | Homo sapiens |