# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Savolitinib (AZD6094) | 28 | Kd apparent | > | 30000 | nM | ALA3991878 | Inactive | nM | Homo sapiens | ||
2. | Dasatinib | 2, BMS-354825 | Kd apparent | > | 30000 | nM | ALA3991878 | Inactive | nM | Homo sapiens | ||
3. | Losmapimod | 10, GW-856553 | Kd apparent | > | 30000 | nM | ALA3991878 | Inactive | nM | Homo sapiens | ||
4. | ALA1614701 | AZD-6244 | Kd apparent | > | 30000 | nM | ALA3991878 | Inactive | nM | Homo sapiens | ||
5. | ALA462018 | TCN-P | Kd apparent | > | 30000 | nM | ALA3991878 | Inactive | nM | Homo sapiens | ||
6. | Poziotinib (HM781-36B) | POZIOTINIB | Kd apparent | > | 30000 | nM | ALA3991878 | Inactive | nM | Homo sapiens | ||
7. | Neratinib (HKI-272) | 25o (table 3) | Kd apparent | > | 30000 | nM | ALA3991878 | Inactive | nM | Homo sapiens | ||
8. | Bafetinib (INNO-406) | 9b | Kd apparent | > | 30000 | nM | ALA3991878 | Inactive | nM | Homo sapiens | ||
9. | Ponatinib (AP24534) | 20g, AP24534 | Kd apparent | > | 30000 | nM | ALA3991878 | Inactive | nM | Homo sapiens | ||
10. | GDC-0941 | 17, GDC-0941 | Kd apparent | > | 30000 | nM | ALA3991878 | Inactive | nM | Homo sapiens | ||
11. | Cerdulatinib (PRT062070) hydrochloride | Cerdulatinib Hydrochloride | Kd apparent | > | 30000 | nM | ALA3991878 | Inactive | nM | Homo sapiens | ||
12. | tesevatinib | TESEVATINIB | Kd apparent | > | 30000 | nM | ALA3991878 | Inactive | nM | Homo sapiens | ||
13. | Ibrutinib (PCI-32765) | SID124898784 | Kd apparent | > | 30000 | nM | ALA3991878 | Inactive | nM | Homo sapiens | ||
14. | AZD5363 | 64, AZD5363 | Kd apparent | > | 30000 | nM | ALA3991878 | Inactive | nM | Homo sapiens | ||
15. | ALA3184679 | AZD-4547 | Kd apparent | > | 30000 | nM | ALA3991878 | Inactive | nM | Homo sapiens | ||
16. | BAY 869766 | REFAMETINIB | Kd apparent | > | 30000 | nM | ALA3991878 | Inactive | nM | Homo sapiens | ||
17. | SAR407899 | 14C | Kd apparent | > | 30000 | nM | ALA3991878 | Inactive | nM | Homo sapiens | ||
18. | Tucatinib (Irbinitinib, ONT-380) | TUCATINIB | Kd apparent | > | 30000 | nM | ALA3991878 | Inactive | nM | Homo sapiens | ||
19. | SU 14813 | SU-14813 | Kd apparent | > | 30000 | nM | ALA3991878 | Inactive | nM | Homo sapiens | ||
20. | BI 2536 | 1 | Kd apparent | > | 30000 | nM | ALA3991878 | Inactive | nM | Homo sapiens |