# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | TG 100801 | 12, TG100801 | Kd apparent | > | 30000 | nM | ALA3991607 | Inactive | nM | Homo sapiens | ||
2. | AZD8931 (Sapitinib) | 2, AZD8931 | Kd apparent | > | 30000 | nM | ALA3991607 | Inactive | nM | Homo sapiens | ||
3. | Regorafenib (BAY 73-4506) | 2, BAY-734506 | Kd apparent | > | 30000 | nM | ALA3991607 | Inactive | nM | Homo sapiens | ||
4. | CEP-32496 | 40, CEP-32496 | Kd apparent | > | 30000 | nM | ALA3991607 | Inactive | nM | Homo sapiens | ||
5. | Crenolanib (CP-868596) | CRENOLANIB | Kd apparent | > | 30000 | nM | ALA3991607 | Inactive | nM | Homo sapiens | ||
6. | K-252a | 2 (K-252a) | Kd apparent | > | 30000 | nM | ALA3991607 | Inactive | nM | Homo sapiens | ||
7. | XL147 | SID174006505 | Kd apparent | > | 30000 | nM | ALA3991607 | Inactive | nM | Homo sapiens | ||
8. | ALA1950289 | 1, CC-930 | Kd apparent | > | 30000 | nM | ALA3991607 | Inactive | nM | Homo sapiens | ||
9. | Decernotinib (VX-509) | DECERNOTINIB | Kd apparent | > | 30000 | nM | ALA3991607 | Inactive | nM | Homo sapiens | ||
10. | ripasudil | ripasudil | Kd apparent | > | 30000 | nM | ALA3991607 | Inactive | nM | Homo sapiens | ||
11. | BYL719 | 8, NVP-BYL719 | Kd apparent | > | 30000 | nM | ALA3991607 | Inactive | nM | Homo sapiens | ||
12. | Axitinib | AG-13736 | Kd apparent | > | 30000 | nM | ALA3991607 | Inactive | nM | Homo sapiens | ||
13. | MK-8776 (SCH 900776) | 29 | Kd apparent | > | 30000 | nM | ALA3991607 | Inactive | nM | Homo sapiens | ||
14. | PF-3758309 | 1, PF-3758309 | Kd apparent | > | 30000 | nM | ALA3991607 | Inactive | nM | Homo sapiens | ||
15. | CX-4945 (Silmitasertib) | 25n | Kd apparent | > | 30000 | nM | ALA3991607 | Inactive | nM | Homo sapiens | ||
16. | Ulixertinib (BVD-523) | ULIXERTINIB | Kd apparent | > | 30000 | nM | ALA3991607 | Inactive | nM | Homo sapiens | ||
17. | Tideglusib | TIDEGLUSIB | Kd apparent | > | 30000 | nM | ALA3991607 | Inactive | nM | Homo sapiens | ||
18. | AZD8055 | 10, AZD-8055 | Kd apparent | > | 30000 | nM | ALA3991607 | Inactive | nM | Homo sapiens | ||
19. | VX-702 | 5, VX-702 | Kd apparent | > | 30000 | nM | ALA3991607 | Inactive | nM | Homo sapiens | ||
20. | Apatinib | SID124955476 | Kd apparent | > | 30000 | nM | ALA3991607 | Inactive | nM | Homo sapiens |