# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BAW2881(NVP-BAW2881) | 2 | IC50 | = | 0.42 | uM | ALA5252744 | 6.38 | nM | Homo sapiens | ||
2. | ALA5288744 | 9 | IC50 | = | 0.05 | uM | ALA5252744 | 7.30 | nM | Homo sapiens | ||
3. | BFH772 | 1 | IC50 | = | 1.1 | uM | ALA5252744 | 5.96 | nM | Homo sapiens | ||
4. | ALA5276611 | 4 | IC50 | = | 0.177 | uM | ALA5252744 | 6.75 | nM | Homo sapiens | ||
5. | ALA5280119 | 10 | IC50 | = | 0.235 | uM | ALA5252744 | 6.63 | nM | Homo sapiens | ||
6. | Vatalanib succinate | CGP-79787D | IC50 | = | 0.064 | uM | ALA5252744 | 7.19 | nM | Homo sapiens | ||
7. | AAL 993 | 5 | IC50 | = | 0.018 | uM | ALA5252744 | 7.75 | nM | Homo sapiens | ||
8. | MnTMPyP pentachloride | 5 | IC50 | = | 0.245 | uM | ALA5252744 | 6.61 | nM | Homo sapiens | ||
9. | Sunitinib | 12b | IC50 | = | 0.024 | uM | ALA5252744 | 7.62 | nM | Homo sapiens | ||
10. | ALA2220486 | LUCITANIB | IC50 | = | 10 | nM | ALA5241428 | 8.00 | nM | Homo sapiens | ||
11. | ALA522892 | 5 | IC50 | = | 8 | nM | ALA5241418 | 8.10 | nM | Homo sapiens | ||
12. | ODM-203 | BDBM247327 | IC50 | = | 5 | nM | ALA5241395 | 8.30 | nM | Homo sapiens | ||
13. | MnTMPyP pentachloride | 5 | IC50 | = | 90 | nM | ALA5241257 | 7.05 | nM | Homo sapiens | ||
14. | 4-Ethyl-N-(4-(1-(tetrahydro-2H-pyran-4-yl)-1H-pyrrolo[2,3-c]pyridin-3-yl)pyridin-2-yl)piperazine-1-carboxamide | 13g; GNF2133 | INH | = | 90 | % | ALA5235860 | % | Homo sapiens | |||
15. | GW843682X | 2 | % of control | = | 1.4 | % | ALA5213212 | % | Homo sapiens | |||
16. | GSK1070916 | GSK-1070916 | IC50 | = | 74 | nM | ALA5213116 | 7.13 | nM | Homo sapiens | ||
17. | Filgotinib (GLPG0634) | SID174006711 | IC50 | = | 274 | nM | ALA5212901 | 6.56 | nM | Homo sapiens | ||
18. | BMS-777607 | 10, BMS-777607 | % of control | = | 0.85 | % | ALA5212890 | % | Homo sapiens | |||
19. | BAY 826 | EUB0000713 | IC50 | = | 0.44 | uM | ALA5213466 | 6.36 | nM | Homo sapiens | ||
20. | ALA5175977 | 28 | IC50 | > | 10 | uM | ALA5165270 | nM | Homo sapiens |