| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5169393 | 11 | INH | = | 66 | % | ALA5157126 | % | Homo sapiens | |||
| 2. |  ALA4455923 | 48c | INH | < | 50 | % | ALA4405370 | % | Homo sapiens | |||
| 3. |  ALA4750196 | 6g | Activity | = | 102.12 | % | ALA4721087 | % | Homo sapiens | |||
| 4. |  Staurosporine | 1 (Staurosporine) | IC50 | = | 1.74 | 10^-8M | ALA4720735 | 7.76 | nM | Homo sapiens | ||
| 5. | Staurosporine | 1 (Staurosporine) | IC50 | = | 6.58 | 10'-8M | ALA4328415 | 7.18 | nM | Homo sapiens | ||
| 6. | Staurosporine | 1 (Staurosporine) | Activity | < | 65 | % | ALA4328051 | % | Homo sapiens | |||
| 7. |  ALA4446405 | 7b; ASR352 | Activity | = | 94.51 | % | ALA4327691 | % | Homo sapiens | |||
| 8. |  ALA4438024 | 7a; NSC30049; NSC49L | Activity | = | 92.63 | % | ALA4327691 | % | Homo sapiens | |||
| 9. |  ALA4749141 | 44 | Activity | = | 90.92 | % | ALA4674386 | % | Homo sapiens | |||
| 10. |  ALA4785602 | 46 | Activity | = | 96.97 | % | ALA4674386 | % | Homo sapiens | |||
| 11. |  BI 605906 | BI605906 | % Ctrl | 102 | % | ALA4887273 | Not Active | % | Homo sapiens | |||
| 12. |  Pelitinib | EKB-569 | Kd apparent | > | 30000 | nM | ALA3991711 | Inactive | nM | Homo sapiens | ||
| 13. |  Ulixertinib (BVD-523) | ULIXERTINIB | Kd apparent | > | 30000 | nM | ALA3991711 | Inactive | nM | Homo sapiens | ||
| 14. |  AT9283 | 16, AT9283 | Kd apparent | > | 30000 | nM | ALA3991711 | Inactive | nM | Homo sapiens | ||
| 15. |  CH5183284 (Debio-1347) | 8; CH5183284; Debio 1347 | Kd apparent | > | 30000 | nM | ALA3991711 | Inactive | nM | Homo sapiens | ||
| 16. |  Filgotinib (GLPG0634) | SID174006711 | Kd apparent | > | 30000 | nM | ALA3991711 | Inactive | nM | Homo sapiens | ||
| 17. |  AZD2014 | 21, AZD2014 | Kd apparent | > | 30000 | nM | ALA3991711 | Inactive | nM | Homo sapiens | ||
| 18. |  Vemurafenib (PLX4032, RG7204) | VEMURAFENIB | Kd apparent | > | 30000 | nM | ALA3991711 | Inactive | nM | Homo sapiens | ||
| 19. |  CX-4945 (Silmitasertib) | 25n | Kd apparent | > | 30000 | nM | ALA3991711 | Inactive | nM | Homo sapiens | ||
| 20. |  TAK-733 | 17, TAK-733 | Kd apparent | > | 30000 | nM | ALA3991711 | Inactive | nM | Homo sapiens |
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