# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Bafetinib (INNO-406) | 9b | Kd apparent | > | 30000 | nM | ALA3991860 | Inactive | nM | Homo sapiens | ||
2. | BMS-690514 | BMS-690514 | Kd apparent | = | 1388 | nM | ALA3991860 | 5.86 | Active | nM | Homo sapiens | |
3. | LY2157299 | GALUNISERTIB | Kd apparent | > | 30000 | nM | ALA3991860 | Inactive | nM | Homo sapiens | ||
4. | Varlitinib | VARLITINIB | Kd apparent | > | 30000 | nM | ALA3991860 | Inactive | nM | Homo sapiens | ||
5. | JANEX-1 | JANEX-1 | Kd apparent | = | 1542 | nM | ALA3991860 | 5.81 | Active | nM | Homo sapiens | |
6. | ripasudil | ripasudil | Kd apparent | > | 30000 | nM | ALA3991860 | Inactive | nM | Homo sapiens | ||
7. | SCIO 469 hydrochloride | SCIO-469 | Kd apparent | > | 30000 | nM | ALA3991860 | Inactive | nM | Homo sapiens | ||
8. | ALA608533 | PKC-412 | Kd apparent | = | 293 | nM | ALA3991860 | 6.53 | Active | nM | Homo sapiens | |
9. | GSK2636771 | SID174006492 | Kd apparent | > | 30000 | nM | ALA3991860 | Inactive | nM | Homo sapiens | ||
10. | AC480 (BMS-599626) | 13, BMS-599626 | Kd apparent | > | 30000 | nM | ALA3991860 | Inactive | nM | Homo sapiens | ||
11. | AMG-208 | 4 | Kd apparent | > | 30000 | nM | ALA3991860 | Inactive | nM | Homo sapiens | ||
12. | MK-1775 | SID103905025 | Kd apparent | > | 30000 | nM | ALA3991860 | Inactive | nM | Homo sapiens | ||
13. | Cobimetinib | 1, XL518, GDC-0973 | Kd apparent | > | 30000 | nM | ALA3991860 | Inactive | nM | Homo sapiens | ||
14. | LY2584702 | LY-2584702 | Kd apparent | > | 30000 | nM | ALA3991860 | Inactive | nM | Homo sapiens | ||
15. | HMN-214 | HMN-214 | Kd apparent | > | 30000 | nM | ALA3991860 | Inactive | nM | Homo sapiens | ||
16. | LY2801653 | MERESTINIB | Kd apparent | > | 30000 | nM | ALA3991860 | Inactive | nM | Homo sapiens | ||
17. | AMG-900 | SID137275938 | Kd apparent | = | 3556 | nM | ALA3991860 | 5.45 | Active | nM | Homo sapiens | |
18. | Afatinib | BIBW-2992 | Kd apparent | > | 30000 | nM | ALA3991860 | Inactive | nM | Homo sapiens | ||
19. | Erlotinib | Tarceva | Kd apparent | > | 30000 | nM | ALA3991860 | Inactive | nM | Homo sapiens | ||
20. | BI 2536 | 1 | Kd apparent | > | 30000 | nM | ALA3991860 | Inactive | nM | Homo sapiens |