# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Savolitinib (AZD6094) | 28 | Kd apparent | > | 30000 | nM | ALA3991889 | Inactive | nM | Homo sapiens | ||
2. | Voxtalisib (XL765) | VOXTALISIB | Kd apparent | > | 30000 | nM | ALA3991889 | Inactive | nM | Homo sapiens | ||
3. | Fostamatinib (R788) | FOSTAMATINIB | Kd apparent | > | 30000 | nM | ALA3991889 | Inactive | nM | Homo sapiens | ||
4. | Tucatinib (Irbinitinib, ONT-380) | TUCATINIB | Kd apparent | > | 30000 | nM | ALA3991889 | Inactive | nM | Homo sapiens | ||
5. | ASP3026 | ASP-3026 | Kd apparent | > | 30000 | nM | ALA3991889 | Inactive | nM | Homo sapiens | ||
6. | Everolimus | EVEROLIMUS | Kd apparent | > | 30000 | nM | ALA3991889 | Inactive | nM | Homo sapiens | ||
7. | DCC-2036 (Rebastinib) | REBASTINIB | Kd apparent | > | 30000 | nM | ALA3991889 | Inactive | nM | Homo sapiens | ||
8. | OSI-930 | OSI-930 | Kd apparent | > | 30000 | nM | ALA3991889 | Inactive | nM | Homo sapiens | ||
9. | JNJ-38877605 | SID137276033 | Kd apparent | > | 30000 | nM | ALA3991889 | Inactive | nM | Homo sapiens | ||
10. | MK-2206 | 17 | Kd apparent | > | 30000 | nM | ALA3991889 | Inactive | nM | Homo sapiens | ||
11. | PDGFR Tyrosine Kinase Inhibitor VI, SU6668 | 5b | Kd apparent | > | 30000 | nM | ALA3991889 | Inactive | nM | Homo sapiens | ||
12. | Trametinib (GSK1120212) | TRAMETINIB | Kd apparent | > | 30000 | nM | ALA3991889 | Inactive | nM | Homo sapiens | ||
13. | Ribociclib | RIBOCICLIB | Kd apparent | > | 30000 | nM | ALA3991889 | Inactive | nM | Homo sapiens | ||
14. | CYT387 | 28 | Kd apparent | > | 30000 | nM | ALA3991889 | Inactive | nM | Homo sapiens | ||
15. | Losmapimod | 10, GW-856553 | Kd apparent | > | 30000 | nM | ALA3991889 | Inactive | nM | Homo sapiens | ||
16. | Dinaciclib (SCH727965) | DINACICLIB | Kd apparent | > | 30000 | nM | ALA3991889 | Inactive | nM | Homo sapiens | ||
17. | X-376 | 2, X376 | Kd apparent | > | 30000 | nM | ALA3991889 | Inactive | nM | Homo sapiens | ||
18. | Afatinib | BIBW-2992 | Kd apparent | > | 30000 | nM | ALA3991889 | Inactive | nM | Homo sapiens | ||
19. | Vandetanib | 22 | Kd apparent | > | 30000 | nM | ALA3991889 | Inactive | nM | Homo sapiens | ||
20. | AMG-208 | 4 | Kd apparent | > | 30000 | nM | ALA3991889 | Inactive | nM | Homo sapiens |