# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | CH4987655 | 24, CH4987655 | Kd apparent | > | 30000 | nM | ALA3991796 | Inactive | nM | Homo sapiens | ||
2. | BI 2536 | 1 | Kd apparent | > | 30000 | nM | ALA3991796 | Inactive | nM | Homo sapiens | ||
3. | CP-547632 | 1 | Kd apparent | > | 30000 | nM | ALA3991796 | Inactive | nM | Homo sapiens | ||
4. | MK-2206 | 17 | Kd apparent | > | 30000 | nM | ALA3991796 | Inactive | nM | Homo sapiens | ||
5. | TAK-593 | 24, TAK-593 | Kd apparent | > | 30000 | nM | ALA3991796 | Inactive | nM | Homo sapiens | ||
6. | LY2603618 | RABUSERTIB | Kd apparent | > | 30000 | nM | ALA3991796 | Inactive | nM | Homo sapiens | ||
7. | LDK378 | 6, LDK378 | Kd apparent | > | 30000 | nM | ALA3991796 | Inactive | nM | Homo sapiens | ||
8. | AZD7762 | AZD-7762 | Kd apparent | > | 30000 | nM | ALA3991796 | Inactive | nM | Homo sapiens | ||
9. | Erlotinib | Tarceva | Kd apparent | > | 30000 | nM | ALA3991796 | Inactive | nM | Homo sapiens | ||
10. | PDGFR Tyrosine Kinase Inhibitor VI, SU6668 | 5b | Kd apparent | = | 1240 | nM | ALA3991796 | 5.91 | Uncertain | nM | Homo sapiens | |
11. | IMD 0354 | TCMDC-125465 | Kd apparent | > | 30000 | nM | ALA3991796 | Inactive | nM | Homo sapiens | ||
12. | glesatinib | MGCD265 | Kd apparent | > | 30000 | nM | ALA3991796 | Inactive | nM | Homo sapiens | ||
13. | Cobimetinib | 1, XL518, GDC-0973 | Kd apparent | > | 30000 | nM | ALA3991796 | Inactive | nM | Homo sapiens | ||
14. | Ribociclib | RIBOCICLIB | Kd apparent | > | 30000 | nM | ALA3991796 | Inactive | nM | Homo sapiens | ||
15. | omipalisib | SID137275909 | Kd apparent | > | 30000 | nM | ALA3991796 | Inactive | nM | Homo sapiens | ||
16. | Gilteritinib | GILTERITINIB | Kd apparent | > | 30000 | nM | ALA3991796 | Inactive | nM | Homo sapiens | ||
17. | 7-(3-(azetidin-1-yl)cyclobutyl)-5-(3-(benzyloxy)phenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine | 15, NVP-AEW541 | Kd apparent | > | 30000 | nM | ALA3991796 | Inactive | nM | Homo sapiens | ||
18. | MK-1775 | SID103905025 | Kd apparent | > | 30000 | nM | ALA3991796 | Inactive | nM | Homo sapiens | ||
19. | CEP-32496 | 40, CEP-32496 | Kd apparent | > | 30000 | nM | ALA3991796 | Inactive | nM | Homo sapiens | ||
20. | Brivanib (BMS-540215) | 12 | Kd apparent | > | 30000 | nM | ALA3991796 | Inactive | nM | Homo sapiens |