# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | K-252a | 2 (K-252a) | Kd apparent | > | 30000 | nM | ALA3991713 | Inactive | nM | Homo sapiens | ||
2. | BYL719 | 8, NVP-BYL719 | Kd apparent | > | 30000 | nM | ALA3991713 | Inactive | nM | Homo sapiens | ||
3. | Entrectinib | SID103905026 | Kd apparent | > | 30000 | nM | ALA3991713 | Inactive | nM | Homo sapiens | ||
4. | RGB-286638 | RGB-286638 | Kd apparent | > | 30000 | nM | ALA3991713 | Inactive | nM | Homo sapiens | ||
5. | Temsirolimus (CCI-779, NSC 683864) | Temsirolimus | Kd apparent | > | 30000 | nM | ALA3991713 | Inactive | nM | Homo sapiens | ||
6. | Ribociclib | RIBOCICLIB | Kd apparent | > | 30000 | nM | ALA3991713 | Inactive | nM | Homo sapiens | ||
7. | ripasudil | ripasudil | Kd apparent | > | 30000 | nM | ALA3991713 | Inactive | nM | Homo sapiens | ||
8. | ALA1094408 | 49 | Kd apparent | > | 30000 | nM | ALA3991713 | Inactive | nM | Homo sapiens | ||
9. | AT13148 | AT-13148 | Kd apparent | > | 30000 | nM | ALA3991713 | Inactive | nM | Homo sapiens | ||
10. | Dabrafenib | 7, GSK2118436 | Kd apparent | > | 30000 | nM | ALA3991713 | Inactive | nM | Homo sapiens | ||
11. | Trametinib (GSK1120212) | TRAMETINIB | Kd apparent | > | 30000 | nM | ALA3991713 | Inactive | nM | Homo sapiens | ||
12. | Cediranib | 5, ZD-2171 | Kd apparent | > | 30000 | nM | ALA3991713 | Inactive | nM | Homo sapiens | ||
13. | Lenvatinib (E7080) | E7080 | Kd apparent | > | 30000 | nM | ALA3991713 | Inactive | nM | Homo sapiens | ||
14. | Defactinib | DEFACTINIB | Kd apparent | > | 30000 | nM | ALA3991713 | Inactive | nM | Homo sapiens | ||
15. | BMS 911543 | BMS-911543 | Kd apparent | > | 30000 | nM | ALA3991713 | Inactive | nM | Homo sapiens | ||
16. | Telatinib | BAY-579352 | Kd apparent | > | 30000 | nM | ALA3991713 | Inactive | nM | Homo sapiens | ||
17. | AZD6482 | AZD-6482 | Kd apparent | > | 30000 | nM | ALA3991713 | Inactive | nM | Homo sapiens | ||
18. | CUDC-101 | 8, CDUC-101 | Kd apparent | > | 30000 | nM | ALA3991713 | Inactive | nM | Homo sapiens | ||
19. | Pelitinib | EKB-569 | Kd apparent | > | 30000 | nM | ALA3991713 | Inactive | nM | Homo sapiens | ||
20. | CH5183284 (Debio-1347) | 8; CH5183284; Debio 1347 | Kd apparent | > | 30000 | nM | ALA3991713 | Inactive | nM | Homo sapiens |