# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4092701 | 12 | IC50 | = | 5.3 | uM | ALA4017288 | 5.28 | nM | Homo sapiens | ||
2. | ALA4066070 | 11 | deltaTm | = | 1.3 | degrees C | ALA4017294 | degrees C | Homo sapiens | |||
3. | ALA4066070 | 11 | deltaTm | = | 2.3 | degrees C | ALA4017293 | degrees C | Homo sapiens | |||
4. | ALA4066070 | 11 | IC50 | = | 4.2 | uM | ALA4017288 | 5.38 | nM | Homo sapiens | ||
5. | ALA4066070 | 11 | INH | 0 | ALA4017287 | Active | % | Homo sapiens | ||||
6. | ALA4066070 | 11 | INH | 0 | ALA4017286 | Active | % | Homo sapiens | ||||
7. | ALA4061514 | 10 | INH | 0 | ALA4017300 | Not Active | % | Homo sapiens | ||||
8. | ALA4061514 | 10 | IC50 | = | 58 | uM | ALA4017288 | 4.24 | nM | Homo sapiens | ||
9. | Brr2 Inhibitor C9 | 9 | INH | 0 | ALA4017299 | Dose-dependent effect | % | Homo sapiens | ||||
10. | Brr2 Inhibitor C9 | 9 | IC50 | = | 1.3 | uM | ALA4017299 | 5.89 | nM | Homo sapiens | ||
11. | Brr2 Inhibitor C9 | 9 | INH | 0 | ALA4017298 | Active | % | Homo sapiens | ||||
12. | Brr2 Inhibitor C9 | 9 | INH | 0 | ALA4017297 | Active | % | Homo sapiens | ||||
13. | Brr2 Inhibitor C9 | 9 | IC50 | = | 0.079 | uM | ALA4017288 | 7.10 | nM | Homo sapiens | ||
14. | ALA4097764 | 8 | IC50 | = | 0.18 | uM | ALA4017288 | 6.75 | nM | Homo sapiens | ||
15. | ALA4070179 | 7 | IC50 | = | 1.4 | uM | ALA4017288 | 5.85 | nM | Homo sapiens | ||
16. | ALA4065018 | 6 | IC50 | = | 0.79 | uM | ALA4017288 | 6.10 | nM | Homo sapiens | ||
17. | ALA4060106 | 5 | IC50 | = | 1.7 | uM | ALA4017288 | 5.77 | nM | Homo sapiens | ||
18. | ALA4074763 | 4 | IC50 | > | 100 | uM | ALA4017288 | nM | Homo sapiens | |||
19. | ALA4087449 | 3 | IC50 | = | 5.3 | uM | ALA4017288 | 5.28 | nM | Homo sapiens | ||
20. | ALA4102900 | 2 | IC50 | > | 100 | uM | ALA4017288 | nM | Homo sapiens |